Detalhe da pesquisa
1.
UV-Induced 1,3,4-Oxadiazole Formation from 5-Substituted Tetrazoles and Carboxylic Acids in Flow.
Chemistry
; 26(65): 14866-14870, 2020 Nov 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-32786060
2.
A high-throughput MALDI-TOF MS biochemical screen for small molecule inhibitors of the antigen aminopeptidase ERAP1.
SLAS Discov
; 28(1): 3-11, 2023 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-36414185
3.
In vivo activity of an azole series of CCR2 antagonists.
Bioorg Med Chem Lett
; 22(23): 7252-5, 2012 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23079519
4.
Identification of a sulfonamide series of CCR2 antagonists.
Bioorg Med Chem Lett
; 20(13): 3961-4, 2010 Jul 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20627722
5.
Author Correction: The mTORC1/4E-BP1 axis represents a critical signaling node during fibrogenesis.
Nat Commun
; 11(1): 4680, 2020 Sep 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-32917879
6.
Discovery of 3-Oxabicyclo[4.1.0]heptane, a Non-nitrogen Containing Morpholine Isostere, and Its Application in Novel Inhibitors of the PI3K-AKT-mTOR Pathway.
J Med Chem
; 62(15): 6972-6984, 2019 08 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-31283227
7.
The mTORC1/4E-BP1 axis represents a critical signaling node during fibrogenesis.
Nat Commun
; 10(1): 6, 2019 01 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-30602778
8.
The discovery of GSK221149A: a potent and selective oxytocin antagonist.
Bioorg Med Chem Lett
; 18(1): 90-4, 2008 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-18032036
9.
Discovery of Potent, Efficient, and Selective Inhibitors of Phosphoinositide 3-Kinase δ through a Deconstruction and Regrowth Approach.
J Med Chem
; 61(24): 11061-11073, 2018 12 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-30532965
10.
Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease.
J Med Chem
; 59(15): 7239-51, 2016 08 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-27429068
11.
Correction to Discovery of 3-Oxabicyclo[4.1.0]heptane, a Non-nitrogen Containing Morpholine Isostere, and Its Application in Novel Inhibitors of the PI3K-AKT-mTOR Pathway.
J Med Chem
; 62(19): 8880, 2019 Oct 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-31553183
12.
Pyridyl-2,5-diketopiperazines as potent, selective, and orally bioavailable oxytocin antagonists: synthesis, pharmacokinetics, and in vivo potency.
J Med Chem
; 55(2): 783-96, 2012 Jan 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-22239250
13.
Three groups good, four groups bad? Atropisomerism in ortho-substituted diaryl ethers.
Angew Chem Int Ed Engl
; 45(35): 5803-7, 2006 Sep 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-16874829
14.
Correction to Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease.
J Med Chem
; 59(20): 9574, 2016 10 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-27726364
15.
Correction to Evolution of a Novel, Orally Bioavailable Series of PI3Kδ Inhibitors from an Inhaled Lead for the Treatment of Respiratory Disease.
J Med Chem
; 59(17): 8148, 2016 09 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-27548024
16.
Investigation of bradykinin metabolism in human and rat plasma in the presence of the dual ACE/NEP inhibitors GW660511X and omapatrilat.
J Pept Sci
; 8(11): 591-600, 2002 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-12487427