Detalhe da pesquisa
1.
Deep Transfer Learning-Based Approach for Glucose Transporter-1 (GLUT1) Expression Assessment.
J Digit Imaging
; 36(6): 2367-2381, 2023 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-37670181
2.
In vitro radiosensitization of breast cancer with hypoxia-activated prodrugs.
J Cell Mol Med
; 26(16): 4577-4590, 2022 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-35841287
3.
Cytochrome P450 Binding and Bioactivation of Tumor-Targeted Duocarmycin Agents.
Drug Metab Dispos
; 50(1): 49-57, 2022 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-34607808
4.
Genetic variation in the ADIPOQ gene and serum adiponectin increase the risk of bladder cancer.
J Appl Biomed
; 20(3): 106-113, 2022 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-36218131
5.
Probing cytochrome P450 (CYP) bioactivation with chloromethylindoline bioprecursors derived from the duocarmycin family of compounds.
Bioorg Med Chem
; 40: 116167, 2021 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-33932713
6.
Design, Synthesis, Biological Evaluation and In Silico Study of Benzyloxybenzaldehyde Derivatives as Selective ALDH1A3 Inhibitors.
Molecules
; 26(19)2021 Sep 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-34641313
7.
Probing cytochrome P450 bioactivation and fluorescent properties with morpholinyl-tethered anthraquinones.
Bioorg Med Chem Lett
; 28(8): 1274-1277, 2018 05 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29576510
8.
Synthesis and biological properties of aryl methyl sulfones.
Bioorg Med Chem
; 26(14): 4113-4126, 2018 08 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-29980364
9.
Therapeutic antibodies against cancer stem cells: a promising approach.
Cancer Immunol Immunother
; 66(11): 1383-1398, 2017 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-28840297
10.
Solid-Phase Synthesis of Duocarmycin Analogues and the Effect of C-Terminal Substitution on Biological Activity.
J Org Chem
; 80(19): 9454-67, 2015 Oct 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-26356089
11.
Quantitative analysis of cytochrome P450 isoforms in human liver microsomes by the combination of proteomics and chemical probe-based assay.
Proteomics
; 14(16): 1943-51, 2014 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-24920405
12.
The Capacity of Drug-Metabolising Enzymes in Modulating the Therapeutic Efficacy of Drugs to Treat Rhabdomyosarcoma.
Cancers (Basel)
; 16(5)2024 Feb 29.
Artigo
em Inglês
| MEDLINE | ID: mdl-38473371
13.
Insight into the liposomal encapsulation of mono and bis-naphthalimides.
RSC Pharm
; 1(2): 272-282, 2024 Jun 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-38899150
14.
Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer.
Eur J Med Chem
; 268: 116193, 2024 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-38364714
15.
Kinetic analysis of intracellular Hoechst 33342--DNA interactions by flow cytometry: misinterpretation of side population status?
Cytometry A
; 83(1): 161-9, 2013 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-23136081
16.
Synthesis and biological evaluation of colchicine C-ring analogues tethered with aliphatic linkers suitable for prodrug derivatisation.
Bioorg Med Chem Lett
; 22(24): 7693-6, 2012 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23103097
17.
The Chemerin-CMKLR1 Axis is Functionally important for Central Regulation of Energy Homeostasis.
Front Physiol
; 13: 897105, 2022.
Artigo
em Inglês
| MEDLINE | ID: mdl-35711300
18.
New aldo-keto reductase 1C3 (AKR1C3) inhibitors based on the hydroxytriazole scaffold.
Eur J Med Chem
; 237: 114366, 2022 Jul 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-35447434
19.
Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer.
J Med Chem
; 65(5): 3833-3848, 2022 03 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-35212533
20.
How can the potential of the duocarmycins be unlocked for cancer therapy?
Drug Discov Today
; 26(2): 577-584, 2021 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-33232841