Detalhe da pesquisa
1.
C-H activation reactions as useful tools for medicinal chemists.
Bioorg Med Chem Lett
; 26(22): 5378-5383, 2016 11 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27765505
2.
Antagonists of the kappa opioid receptor.
Bioorg Med Chem Lett
; 24(9): 2021-32, 2014 May 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24690494
3.
Modulators of the Sphingosine 1-phosphate receptor 1.
Bioorg Med Chem Lett
; 23(23): 6377-89, 2013 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24125884
4.
SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists.
Bioorg Med Chem Lett
; 23(3): 614-9, 2013 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23287738
5.
Discovery, design and synthesis of a selective S1P(3) receptor allosteric agonist.
Bioorg Med Chem Lett
; 23(23): 6346-9, 2013 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24135724
6.
Discovery, design and synthesis of novel potent and selective sphingosine-1-phosphate 4 receptor (S1P4-R) agonists.
Bioorg Med Chem Lett
; 22(1): 537-42, 2012 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22119461
7.
Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7).
Bioorg Med Chem Lett
; 22(23): 7135-41, 2012 Dec 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-23079522
8.
SAR analysis of innovative selective small molecule antagonists of sphingosine-1-phosphate 4 (S1P4) receptor.
Bioorg Med Chem Lett
; 21(18): 5470-4, 2011 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21783362
9.
Discovery, design and synthesis of the first reported potent and selective sphingosine-1-phosphate 4 (S1P4) receptor antagonists.
Bioorg Med Chem Lett
; 21(12): 3632-6, 2011 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21570287
10.
Discovery, synthesis and SAR analysis of novel selective small molecule S1P4-R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chemotype.
Bioorg Med Chem Lett
; 21(22): 6739-45, 2011 Nov 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21982495
11.
Identification of a potent and selective σ1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells.
Bioorg Med Chem
; 19(21): 6210-24, 2011 Nov 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21967807
12.
Design, synthesis and SAR analysis of novel selective sigma1 ligands (Part 2).
Bioorg Med Chem
; 18(3): 1204-12, 2010 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-20045339
13.
Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140).
J Med Chem
; 62(4): 1761-1780, 2019 02 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-30707578
14.
Substituted benzylaminoalkylindoles with preference for the sigma2 binding site.
Eur J Med Chem
; 43(10): 2073-81, 2008 Oct.
Artigo
em Inglês
| MEDLINE | ID: mdl-18069094
15.
Microwave-assisted extraction of coumarin and related compounds from Melilotus officinalis (L.) Pallas as an alternative to Soxhlet and ultrasound-assisted extraction.
J Chromatogr A
; 1125(2): 147-51, 2006 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-16769080
16.
Sphingosine 1-phosphate receptor 1 agonists: a patent review (2013-2015).
Expert Opin Ther Pat
; 26(4): 455-70, 2016.
Artigo
em Inglês
| MEDLINE | ID: mdl-26947494
17.
Sphingosine 1-phosphate receptor agonists: a patent review (2010-2012).
Expert Opin Ther Pat
; 23(7): 817-41, 2013 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-23541049
18.
Design, synthesis, and SAR analysis of novel selective sigma1 ligands.
Bioorg Med Chem
; 15(2): 771-83, 2007 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-17088069
19.
Highly diastereoselective synthesis of enantiopure naphthylaminoalcohols with analgesic properties.
Chirality
; 18(10): 841-8, 2006 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-16917832
20.
Enantioselective chromatography and absolute configuration of N,N-dimethyl-3-(naphthalen-2-yl)-butan-1-amines: potential sigma1 ligands.
Chirality
; 18(4): 245-53, 2006 May 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-16521084