Detalhe da pesquisa
1.
Identification of small-molecule protein-protein interaction inhibitors for NKG2D.
Proc Natl Acad Sci U S A
; 120(18): e2216342120, 2023 05 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-37098070
2.
Development of small molecule inhibitors of natural killer group 2D receptor (NKG2D).
Bioorg Med Chem Lett
; 96: 129492, 2023 11 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37778428
3.
One-Pot Reductive Alkylation of 2,4-Dihydroxy Quinolines and Pyridines.
J Org Chem
; 86(10): 7148-7162, 2021 05 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-33913727
4.
3-Substituted Quinolines as RORγt Inverse Agonists.
Bioorg Med Chem Lett
; 29(12): 1463-1470, 2019 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31010722
5.
Identification and structure activity relationships of quinoline tertiary alcohol modulators of RORγt.
Bioorg Med Chem Lett
; 27(9): 2047-2057, 2017 05 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28318945
6.
6-Substituted quinolines as RORγt inverse agonists.
Bioorg Med Chem Lett
; 27(23): 5277-5283, 2017 12 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-29079472
7.
Enhanced UV-Irradiated Photocatalytic Degradation of Malachite Green by Porous WO3 Decorated on 2D Graphene Sheet.
Appl Biochem Biotechnol
; 195(6): 3966-3980, 2023 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-35394253
8.
Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible factor prolyl hydroxylase inhibitor.
Mol Pharmacol
; 79(6): 910-20, 2011 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-21372172
9.
Protecting-group-free synthesis of a dual CCK1/CCK2 receptor antagonist.
Org Biomol Chem
; 9(8): 2654-60, 2011 Apr 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-21365101
10.
A one-step synthesis of 2,4-unsubstituted quinoline-3-carboxylic acid esters from o-nitrobenzaldehydes.
J Org Chem
; 75(10): 3488-91, 2010 May 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-20420395
11.
Characterization of a robust enzymatic assay for inhibitors of 2-oxoglutarate-dependent hydroxylases.
J Biomol Screen
; 14(6): 627-35, 2009 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-19498081
12.
Anthranilic sulfonamide CCK1/CCK2 dual receptor antagonists II: tuning of receptor selectivity and in vivo efficacy.
Bioorg Med Chem Lett
; 19(22): 6376-8, 2009 Nov 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-19815410
13.
Beyond Traditional Structure-Based Drug Design: The Role of Iron Complexation, Strain, and Water in the Binding of Inhibitors for Hypoxia-Inducible Factor Prolyl Hydroxylase 2.
ACS Omega
; 4(4): 6703-6708, 2019 Apr 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-31179408
14.
Identification and optimization of anthranilic sulfonamides as novel, selective cholecystokinin-2 receptor antagonists.
J Med Chem
; 49(21): 6371-90, 2006 Oct 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-17034143
15.
Prolyl hydroxylase inhibition corrects functional iron deficiency and inflammation-induced anaemia in rats.
Br J Pharmacol
; 172(16): 4078-88, 2015 Aug.
Artigo
em Inglês
| MEDLINE | ID: mdl-25988595
16.
Improved Utility of Photolabile Solid Phase Synthesis Supports for the Synthesis of Oligonucleotides Containing 3'-Hydroxyl Termini.
J Org Chem
; 61(2): 525-529, 1996 Jan 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-11666970
17.
Benzimidazole-2-pyrazole HIF Prolyl 4-Hydroxylase Inhibitors as Oral Erythropoietin Secretagogues.
ACS Med Chem Lett
; 1(9): 526-9, 2010 Dec 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-24900242
18.
Tetrahydroindazole inhibitors of bacterial type II topoisomerases. Part 2: SAR development and potency against multidrug-resistant strains.
Bioorg Med Chem Lett
; 17(10): 2718-22, 2007 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-17382544
19.
Identification of novel inhibitors of bacterial translation elongation factors.
Antimicrob Agents Chemother
; 49(1): 131-6, 2005 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-15616286
20.
Novel glycine transporter type-2 reuptake inhibitors. Part 1: alpha-amino acid derivatives.
Bioorg Med Chem
; 12(16): 4477-92, 2004 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-15265498