Detalhe da pesquisa
1.
P-Glycoprotein-Mediated Efflux Reduces the In Vivo Efficacy of a Therapeutic Targeting the Gastrointestinal Parasite Cryptosporidium.
J Infect Dis
; 220(7): 1188-1198, 2019 08 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-31180118
2.
Pharmacokinetics and In Vivo Efficacy of Pyrazolopyrimidine, Pyrrolopyrimidine, and 5-Aminopyrazole-4-Carboxamide Bumped Kinase Inhibitors against Toxoplasmosis.
J Infect Dis
; 219(9): 1464-1473, 2019 04 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-30423128
3.
Necessity of Bumped Kinase Inhibitor Gastrointestinal Exposure in Treating Cryptosporidium Infection.
J Infect Dis
; 216(1): 55-63, 2017 07 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28541457
4.
Bumped-Kinase Inhibitors for Cryptosporidiosis Therapy.
J Infect Dis
; 215(8): 1275-1284, 2017 04 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-28329187
5.
Novel Bumped Kinase Inhibitors Are Safe and Effective Therapeutics in the Calf Clinical Model for Cryptosporidiosis.
J Infect Dis
; 214(12): 1856-1864, 2016 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27923949
6.
A novel calcium-dependent protein kinase inhibitor as a lead compound for treating cryptosporidiosis.
J Infect Dis
; 208(8): 1342-8, 2013 Oct 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23878324
7.
Pyrrolopyrimidine Bumped Kinase Inhibitors for the Treatment of Cryptosporidiosis.
ACS Infect Dis
; 7(5): 1200-1207, 2021 05 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-33565854
8.
One health therapeutics: Target-Based drug development for cryptosporidiosis and other apicomplexa diseases.
Vet Parasitol
; 289: 109336, 2021 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-33418437
9.
Bumped Kinase Inhibitors as therapy for apicomplexan parasitic diseases: lessons learned.
Int J Parasitol
; 50(5): 413-422, 2020 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-32224121
10.
Bumped kinase inhibitor 1369 is effective against Cystoisospora suis in vivo and in vitro.
Int J Parasitol Drugs Drug Resist
; 10: 9-19, 2019 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-30959327
11.
In vitro growth inhibition of Theileria equi by bumped kinase inhibitors.
Vet Parasitol
; 251: 90-94, 2018 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-29426483
12.
7 H-Pyrrolo[2,3- d]pyrimidin-4-amine-Based Inhibitors of Calcium-Dependent Protein Kinase 1 Have Distinct Inhibitory and Oral Pharmacokinetic Characteristics Compared with 1 H-Pyrazolo[3,4- d]pyrimidin-4-amine-Based Inhibitors.
ACS Infect Dis
; 4(4): 516-522, 2018 04 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-29522315
13.
Advances in bumped kinase inhibitors for human and animal therapy for cryptosporidiosis.
Int J Parasitol
; 47(12): 753-763, 2017 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-28899690