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Discovery and Characterization of Biased Allosteric Agonists of the Chemokine Receptor CXCR3.
Milanos, Lampros; Brox, Regine; Frank, Theresa; Poklukar, Gasper; Palmisano, Ralf; Waibel, Reiner; Einsiedel, Jürgen; Dürr, Maximilian; Ivanovic-Burmazovic, Ivana; Larsen, Olav; Hjortø, Gertrud Malene; Rosenkilde, Mette Marie; Tschammer, Nuska.
Afiliação
  • Milanos L; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University , Schuhstraße 19, 91052 Erlangen, Germany.
  • Brox R; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University , Schuhstraße 19, 91052 Erlangen, Germany.
  • Frank T; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University , Schuhstraße 19, 91052 Erlangen, Germany.
  • Poklukar G; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University , Schuhstraße 19, 91052 Erlangen, Germany.
  • Palmisano R; Faculty of Pharmacy, University of Ljubljana , Askerceva 7, 1000 Ljubljana, Slovenia.
  • Waibel R; Optical Imaging Center Erlangen, Friedrich Alexander University , Hartmannstraße 14, 91052 Erlangen, Germany.
  • Einsiedel J; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University , Schuhstraße 19, 91052 Erlangen, Germany.
  • Dürr M; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University , Schuhstraße 19, 91052 Erlangen, Germany.
  • Ivanovic-Burmazovic I; Department of Chemistry and Pharmacy, Bioorganic Chemistry, Friedrich Alexander University , Egerlandstraße 1, 91058 Erlangen, Germany.
  • Larsen O; Department of Chemistry and Pharmacy, Bioorganic Chemistry, Friedrich Alexander University , Egerlandstraße 1, 91058 Erlangen, Germany.
  • Hjortø GM; Department of Neuroscience and Pharmacology, Laboratory for Molecular Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen , Blegdamsvej 3B, DK-2200 Copenhagen N, Denmark.
  • Rosenkilde MM; Department of Neuroscience and Pharmacology, Laboratory for Molecular Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen , Blegdamsvej 3B, DK-2200 Copenhagen N, Denmark.
  • Tschammer N; Department of Neuroscience and Pharmacology, Laboratory for Molecular Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen , Blegdamsvej 3B, DK-2200 Copenhagen N, Denmark.
J Med Chem ; 59(5): 2222-43, 2016 Mar 10.
Article em En | MEDLINE | ID: mdl-26862767

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tetra-Hidroisoquinolinas / Regulação Alostérica / Receptores CXCR3 / Descoberta de Drogas Limite: Animals / Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tetra-Hidroisoquinolinas / Regulação Alostérica / Receptores CXCR3 / Descoberta de Drogas Limite: Animals / Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Alemanha