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NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids.
Simeth, Nadja A; Bause, Manuel; Dobmeier, Michael; Kling, Ralf C; Lachmann, Daniel; Hübner, Harald; Einsiedel, Jürgen; Gmeiner, Peter; König, Burkhard.
Afiliação
  • Simeth NA; Faculty of Chemistry and Pharmacy, Institute of Organic Chemistry, University of Regensburg, Universitätsstr. 31, 93053 Regensburg, Germany.
  • Bause M; Faculty of Chemistry and Pharmacy, Institute of Organic Chemistry, University of Regensburg, Universitätsstr. 31, 93053 Regensburg, Germany.
  • Dobmeier M; Faculty of Chemistry and Pharmacy, Institute of Organic Chemistry, University of Regensburg, Universitätsstr. 31, 93053 Regensburg, Germany.
  • Kling RC; Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich-Alexander-Universität Erlangen Nürnberg (FAU), Schuhstr. 19, 91052 Erlangen, Germany; Institute of Physiology, Paracelsus Medical University Nürnberg, 90419 Nürnberg, Germany.
  • Lachmann D; Faculty of Chemistry and Pharmacy, Institute of Organic Chemistry, University of Regensburg, Universitätsstr. 31, 93053 Regensburg, Germany.
  • Hübner H; Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich-Alexander-Universität Erlangen Nürnberg (FAU), Schuhstr. 19, 91052 Erlangen, Germany.
  • Einsiedel J; Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich-Alexander-Universität Erlangen Nürnberg (FAU), Schuhstr. 19, 91052 Erlangen, Germany.
  • Gmeiner P; Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich-Alexander-Universität Erlangen Nürnberg (FAU), Schuhstr. 19, 91052 Erlangen, Germany. Electronic address: peter.gmeiner@fau.de.
  • König B; Faculty of Chemistry and Pharmacy, Institute of Organic Chemistry, University of Regensburg, Universitätsstr. 31, 93053 Regensburg, Germany. Electronic address: burkhard.koenig@ur.de.
Bioorg Med Chem ; 25(1): 350-359, 2017 01 01.
Article em En | MEDLINE | ID: mdl-27842797

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Ácido Pirrolidonocarboxílico / Neurotensina / Receptores de Neurotensina / Peptidomiméticos / Furanos Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Ácido Pirrolidonocarboxílico / Neurotensina / Receptores de Neurotensina / Peptidomiméticos / Furanos Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Alemanha