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Discovery of novel DNA methyltransferase 3A inhibitors via structure-based virtual screening and biological assays.
Shao, Zhiyuan; Xu, Pan; Xu, Wen; Li, Linjuan; Liu, Shien; Zhang, Rukang; Liu, Yu-Chih; Zhang, Chenhua; Chen, Shijie; Luo, Cheng.
Afiliação
  • Shao Z; Nano Science and Technology Institute, University of Science and Technology of China, Suzhou 215123, China.
  • Xu P; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of MateriaMedica, Chinese Academy of Sciences, Shanghai 201203, China.
  • Xu W; Obstetrics & Gynecology Hospital of Fudan University, No. 419 Fangxie Road, Shanghai 200011, China.
  • Li L; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of MateriaMedica, Chinese Academy of Sciences, Shanghai 201203, China; School of Life Science and Technology, Shanghai Tech University, Shanghai 200031, China.
  • Liu S; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of MateriaMedica, Chinese Academy of Sciences, Shanghai 201203, China.
  • Zhang R; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of MateriaMedica, Chinese Academy of Sciences, Shanghai 201203, China; School of Life Science and Technology, Shanghai Tech University, Shanghai 200031, China.
  • Liu YC; Shanghai ChemPartner Co., LTD, Building 5, 998, Halei Road, Zhangjiang Hi-Tech Park, Pudong New Area, Shanghai 201203, China.
  • Zhang C; Shanghai ChemPartner Co., LTD, Building 5, 998, Halei Road, Zhangjiang Hi-Tech Park, Pudong New Area, Shanghai 201203, China.
  • Chen S; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of MateriaMedica, Chinese Academy of Sciences, Shanghai 201203, China. Electronic address: shijiechen@simm.ac.cn.
  • Luo C; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of MateriaMedica, Chinese Academy of Sciences, Shanghai 201203, China. Electronic address: cluo@simm.ac.cn.
Bioorg Med Chem Lett ; 27(2): 342-346, 2017 01 15.
Article em En | MEDLINE | ID: mdl-27899265

Texto completo: 1 Base de dados: MEDLINE Assunto principal: DNA (Citosina-5-)-Metiltransferases / Inibidores Enzimáticos / Descoberta de Drogas Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: China

Texto completo: 1 Base de dados: MEDLINE Assunto principal: DNA (Citosina-5-)-Metiltransferases / Inibidores Enzimáticos / Descoberta de Drogas Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: China