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NMR structure-based optimization of Staphylococcus aureus sortase A pyridazinone inhibitors.
Chan, Albert H; Yi, Sung Wook; Weiner, Ethan M; Amer, Brendan R; Sue, Christopher K; Wereszczynski, Jeff; Dillen, Carly A; Senese, Silvia; Torres, Jorge Z; McCammon, J Andrew; Miller, Lloyd S; Jung, Michael E; Clubb, Robert T.
Afiliação
  • Chan AH; Department of Chemistry and Biochemistry, University of California, Los Angeles, Los Angeles, CA, USA.
  • Yi SW; UCLA-DOE Institute of Genomics and Proteomics, University of California, Los Angeles, Los Angeles, CA, USA.
  • Weiner EM; Molecular Biology Institute, University of California, Los Angeles, Los Angeles, CA, USA.
  • Amer BR; Department of Chemistry and Biochemistry, University of California, Los Angeles, Los Angeles, CA, USA.
  • Sue CK; Department of Chemistry and Biochemistry, University of California, Los Angeles, Los Angeles, CA, USA.
  • Wereszczynski J; UCLA-DOE Institute of Genomics and Proteomics, University of California, Los Angeles, Los Angeles, CA, USA.
  • Dillen CA; Molecular Biology Institute, University of California, Los Angeles, Los Angeles, CA, USA.
  • Senese S; Department of Chemistry and Biochemistry, University of California, Los Angeles, Los Angeles, CA, USA.
  • Torres JZ; UCLA-DOE Institute of Genomics and Proteomics, University of California, Los Angeles, Los Angeles, CA, USA.
  • McCammon JA; Molecular Biology Institute, University of California, Los Angeles, Los Angeles, CA, USA.
  • Miller LS; Department of Chemistry and Biochemistry, University of California, Los Angeles, Los Angeles, CA, USA.
  • Jung ME; Department of Physics and Center for Molecular Study of Condensed Soft Matter, Illinois Institute of Technology, Chicago, IL, USA.
  • Clubb RT; Department of Dermatology, Johns Hopkins University School of Medicine, Baltimore, MD, USA.
Chem Biol Drug Des ; 90(3): 327-344, 2017 Sep.
Article em En | MEDLINE | ID: mdl-28160417

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridazinas / Staphylococcus aureus / Proteínas de Bactérias / Aminoaciltransferases / Inibidores Enzimáticos / Antibacterianos Limite: Humans Idioma: En Revista: Chem Biol Drug Des Assunto da revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridazinas / Staphylococcus aureus / Proteínas de Bactérias / Aminoaciltransferases / Inibidores Enzimáticos / Antibacterianos Limite: Humans Idioma: En Revista: Chem Biol Drug Des Assunto da revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos