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ML290 is a biased allosteric agonist at the relaxin receptor RXFP1.
Kocan, Martina; Sarwar, Mohsin; Ang, Sheng Y; Xiao, Jingbo; Marugan, Juan J; Hossain, Mohammed A; Wang, Chao; Hutchinson, Dana S; Samuel, Chrishan S; Agoulnik, Alexander I; Bathgate, Ross A D; Summers, Roger J.
Afiliação
  • Kocan M; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia. Martina.Kocan@monash.edu.
  • Sarwar M; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.
  • Ang SY; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.
  • Xiao J; Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, USA.
  • Marugan JJ; Preclinical Innovation, National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, USA.
  • Hossain MA; The Florey Institute of Neuroscience and Mental Health, Parkville, Australia.
  • Wang C; Cardiovascular Disease Program, Biomedicine Discovery Institute and Department of Pharmacology, Monash University, Clayton, Australia.
  • Hutchinson DS; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Australia.
  • Samuel CS; Cardiovascular Disease Program, Biomedicine Discovery Institute and Department of Pharmacology, Monash University, Clayton, Australia.
  • Agoulnik AI; Department of Human and Molecular Genetics, Herbert Wertheim College of Medicine, Florida International University, Florida, USA.
  • Bathgate RAD; The Florey Institute of Neuroscience and Mental Health, Parkville, Australia.
  • Summers RJ; Department of Biochemistry and Molecular Biology, University of Melbourne, Parkville, Australia.
Sci Rep ; 7(1): 2968, 2017 06 07.
Article em En | MEDLINE | ID: mdl-28592882

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores de Peptídeos / Receptores Acoplados a Proteínas G Limite: Humans Idioma: En Revista: Sci Rep Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Austrália

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores de Peptídeos / Receptores Acoplados a Proteínas G Limite: Humans Idioma: En Revista: Sci Rep Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Austrália