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Design and Optimization of Benzopiperazines as Potent Inhibitors of BET Bromodomains.
Millan, David S; Kayser-Bricker, Katherine J; Martin, Matthew W; Talbot, Adam C; Schiller, Shawn E R; Herbertz, Torsten; Williams, Grace L; Luke, George P; Hubbs, Stephen; Alvarez Morales, Monica A; Cardillo, Daniel; Troccolo, Paul; Mendes, Rachel L; McKinnon, Crystal.
Afiliação
  • Millan DS; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Kayser-Bricker KJ; FORMA Therapeutics Inc., 35 Northeast Industrial Road, Branford, Connecticut 06405, United States.
  • Martin MW; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Talbot AC; FORMA Therapeutics Inc., 35 Northeast Industrial Road, Branford, Connecticut 06405, United States.
  • Schiller SER; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Herbertz T; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Williams GL; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Luke GP; FORMA Therapeutics Inc., 35 Northeast Industrial Road, Branford, Connecticut 06405, United States.
  • Hubbs S; FORMA Therapeutics Inc., 35 Northeast Industrial Road, Branford, Connecticut 06405, United States.
  • Alvarez Morales MA; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Cardillo D; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Troccolo P; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • Mendes RL; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
  • McKinnon C; FORMA Therapeutics Inc., 500 Arsenal Street, Suite 100, Watertown, Massachusetts 02472, United States.
ACS Med Chem Lett ; 8(8): 847-852, 2017 Aug 10.
Article em En | MEDLINE | ID: mdl-28835800
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Texto completo: 1 Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos