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Identification of an (-)-englerin A analogue, which antagonizes (-)-englerin A at TRPC1/4/5 channels.
Rubaiy, Hussein N; Seitz, Tobias; Hahn, Sven; Choidas, Axel; Habenberger, Peter; Klebl, Bert; Dinkel, Klaus; Nussbaumer, Peter; Waldmann, Herbert; Christmann, Mathias; Beech, David J.
Afiliação
  • Rubaiy HN; School of Medicine, University of Leeds, Leeds, UK.
  • Seitz T; Institute of Chemistry and Biochemistry, Freie Universität Berlin, Berlin, Germany.
  • Hahn S; Institute of Chemistry and Biochemistry, Freie Universität Berlin, Berlin, Germany.
  • Choidas A; Lead Discovery Center GmbH, Dortmund, Germany.
  • Habenberger P; Lead Discovery Center GmbH, Dortmund, Germany.
  • Klebl B; Lead Discovery Center GmbH, Dortmund, Germany.
  • Dinkel K; Lead Discovery Center GmbH, Dortmund, Germany.
  • Nussbaumer P; Lead Discovery Center GmbH, Dortmund, Germany.
  • Waldmann H; Max-Planck-Institut für molekulare Physiologie, Dortmund, Germany.
  • Christmann M; Institute of Chemistry and Biochemistry, Freie Universität Berlin, Berlin, Germany.
  • Beech DJ; School of Medicine, University of Leeds, Leeds, UK.
Br J Pharmacol ; 175(5): 830-839, 2018 03.
Article em En | MEDLINE | ID: mdl-29247460

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sesquiterpenos de Guaiano / Canais de Cátion TRPC / Potenciais da Membrana Tipo de estudo: Diagnostic_studies / Prognostic_studies Limite: Humans Idioma: En Revista: Br J Pharmacol Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Reino Unido

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sesquiterpenos de Guaiano / Canais de Cátion TRPC / Potenciais da Membrana Tipo de estudo: Diagnostic_studies / Prognostic_studies Limite: Humans Idioma: En Revista: Br J Pharmacol Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Reino Unido