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Piperlongumine and some of its analogs inhibit selectively the human immunoproteasome over the constitutive proteasome.
Bosc, Elodie; Nastri, Jhennifer; Lefort, Valérie; Valli, Marilia; Contiguiba, Fernando; Pioli, Renan; Furlan, Maysa; Bolzani, Vanderlan da Silva; El Amri, Chahrazade; Reboud-Ravaux, Michèle.
Afiliação
  • Bosc E; Sorbonne Université, UPMC Univ Paris 06-CNRS, IBPS, UMR 8256, Inserm ERL1164, B2A, 7 Quai Saint Bernard, F75005 Paris, France.
  • Nastri J; Nuclei of Bioassays, Biosynthesis and Ecophysiology of Natural Products (NuBBE), Department of Organic Chemistry, Institute of Chemistry, Sao Paulo State University - UNESP, 14800-060, Araraquara, SP, Brazil.
  • Lefort V; Sorbonne Université, UPMC Univ Paris 06-CNRS, IBPS, UMR 8256, Inserm ERL1164, B2A, 7 Quai Saint Bernard, F75005 Paris, France.
  • Valli M; Nuclei of Bioassays, Biosynthesis and Ecophysiology of Natural Products (NuBBE), Department of Organic Chemistry, Institute of Chemistry, Sao Paulo State University - UNESP, 14800-060, Araraquara, SP, Brazil.
  • Contiguiba F; Institute for Natural Products Research Walter Mors, Health Sciences Center - HSC, Federal University of Rio de Janeiro - UFRJ, 21941902, Rio de Janeiro, RJ, Brazil.
  • Pioli R; Institute of Chemistry, Department of Organic Chemistry, University of São Paulo - USP, 05508-000, São Paulo, SP, Brazil.
  • Furlan M; Nuclei of Bioassays, Biosynthesis and Ecophysiology of Natural Products (NuBBE), Department of Organic Chemistry, Institute of Chemistry, Sao Paulo State University - UNESP, 14800-060, Araraquara, SP, Brazil.
  • Bolzani VDS; Nuclei of Bioassays, Biosynthesis and Ecophysiology of Natural Products (NuBBE), Department of Organic Chemistry, Institute of Chemistry, Sao Paulo State University - UNESP, 14800-060, Araraquara, SP, Brazil.
  • El Amri C; Sorbonne Université, UPMC Univ Paris 06-CNRS, IBPS, UMR 8256, Inserm ERL1164, B2A, 7 Quai Saint Bernard, F75005 Paris, France. Electronic address: chahrazade.el_amri@upmc.fr.
  • Reboud-Ravaux M; Sorbonne Université, UPMC Univ Paris 06-CNRS, IBPS, UMR 8256, Inserm ERL1164, B2A, 7 Quai Saint Bernard, F75005 Paris, France. Electronic address: michele.reboud@upmc.fr.
Biochem Biophys Res Commun ; 496(3): 961-966, 2018 02 12.
Article em En | MEDLINE | ID: mdl-29355526

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Imunoproteínas / Apoptose / Complexo de Endopeptidases do Proteassoma / Dioxolanos Limite: Humans Idioma: En Revista: Biochem Biophys Res Commun Ano de publicação: 2018 Tipo de documento: Article País de afiliação: França

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Imunoproteínas / Apoptose / Complexo de Endopeptidases do Proteassoma / Dioxolanos Limite: Humans Idioma: En Revista: Biochem Biophys Res Commun Ano de publicação: 2018 Tipo de documento: Article País de afiliação: França