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Myc phosphorylation in its basic helix-loop-helix region destabilizes transient α-helical structures, disrupting Max and DNA binding.
Macek, Pavel; Cliff, Matthew J; Embrey, Kevin J; Holdgate, Geoffrey A; Nissink, J Willem M; Panova, Stanislava; Waltho, Jonathan P; Davies, Rick A.
Afiliação
  • Macek P; From AstraZeneca, IMED Discovery Sciences, Alderley Park SK10 4TG, United Kingdom, macek@nmr-bio.com.
  • Cliff MJ; the Manchester Institute of Biotechnology and School of Chemistry, University of Manchester, Manchester M1 7DN, United Kingdom.
  • Embrey KJ; AstraZeneca, IMED Discovery Sciences, Cambridge CB4 0WG, United Kingdom.
  • Holdgate GA; AstraZeneca, IMED Discovery Sciences, Cambridge CB4 0WG, United Kingdom.
  • Nissink JWM; AstraZeneca, IMED Oncology, Cambridge CB4 0WG, United Kingdom, and.
  • Panova S; the Manchester Institute of Biotechnology and School of Chemistry, University of Manchester, Manchester M1 7DN, United Kingdom.
  • Waltho JP; the Manchester Institute of Biotechnology and School of Chemistry, University of Manchester, Manchester M1 7DN, United Kingdom.
  • Davies RA; From AstraZeneca, IMED Discovery Sciences, Alderley Park SK10 4TG, United Kingdom, rick.davies@astrazeneca.com.
J Biol Chem ; 293(24): 9301-9310, 2018 06 15.
Article em En | MEDLINE | ID: mdl-29695509

Texto completo: 1 Base de dados: MEDLINE Assunto principal: DNA / Proteínas Proto-Oncogênicas c-myc / Fatores de Transcrição de Zíper de Leucina e Hélice-Alça-Hélix Básicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: J Biol Chem Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: DNA / Proteínas Proto-Oncogênicas c-myc / Fatores de Transcrição de Zíper de Leucina e Hélice-Alça-Hélix Básicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: J Biol Chem Ano de publicação: 2018 Tipo de documento: Article