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Synthesis, in vitro and in silico evaluation of diaryl heptanones as potential 5LOX enzyme inhibitors.
Meka, Bharani; Ravada, Suryachandra Rao; Muthyala, Murali Krishna Kumar; Kurre, Purna Nagasree; Golakoti, Trimurtulu.
Afiliação
  • Meka B; LailaImpex R&D Center, Unit-I, Phase-III, Jawahar Auto Nagar, Vijayawada 520 007, Andhra Pradesh, India.
  • Ravada SR; LailaImpex R&D Center, Unit-I, Phase-III, Jawahar Auto Nagar, Vijayawada 520 007, Andhra Pradesh, India.
  • Muthyala MKK; Department of Pharmaceutical Chemistry, AU College of Pharmaceutical Sciences, Andhra University, Visakhapatnam 530 003, Andhra Pradesh, India.
  • Kurre PN; Department of Pharmaceutical Chemistry, AU College of Pharmaceutical Sciences, Andhra University, Visakhapatnam 530 003, Andhra Pradesh, India.
  • Golakoti T; LailaImpex R&D Center, Unit-I, Phase-III, Jawahar Auto Nagar, Vijayawada 520 007, Andhra Pradesh, India. Electronic address: research@lailanutra.in.
Bioorg Chem ; 80: 408-421, 2018 10.
Article em En | MEDLINE | ID: mdl-29986187

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Araquidonato 5-Lipoxigenase / Inibidores de Lipoxigenase / Diarileptanoides Limite: Humans Idioma: En Revista: Bioorg Chem Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Araquidonato 5-Lipoxigenase / Inibidores de Lipoxigenase / Diarileptanoides Limite: Humans Idioma: En Revista: Bioorg Chem Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Índia