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Discovery of Potent and Selective Methylenephosphonic Acid CD73 Inhibitors.
Sharif, Ehesan U; Kalisiak, Jaroslaw; Lawson, Kenneth V; Miles, Dillon H; Newcomb, Eric; Lindsey, Erick A; Rosen, Brandon R; Debien, Laurent P P; Chen, Ada; Zhao, Xiaoning; Young, Stephen W; Walker, Nigel P; Sträter, Norbert; Scaletti, Emma R; Jin, Lixia; Xu, Guifen; Leleti, Manmohan R; Powers, Jay P.
Afiliação
  • Sharif EU; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Kalisiak J; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Lawson KV; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Miles DH; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Newcomb E; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Lindsey EA; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Rosen BR; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Debien LPP; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Chen A; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Zhao X; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Young SW; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Walker NP; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Sträter N; Institute of Bioanalytical Chemistry, Center for Biotechnology and Biomedicine, Leipzig University, Deutscher Platz 5, D-04103 Leipzig, Germany.
  • Scaletti ER; Institute of Bioanalytical Chemistry, Center for Biotechnology and Biomedicine, Leipzig University, Deutscher Platz 5, D-04103 Leipzig, Germany.
  • Jin L; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Xu G; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Leleti MR; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
  • Powers JP; Arcus Biosciences, Inc., 3928 Point Eden Way, Hayward, California 94545, United States.
J Med Chem ; 64(1): 845-860, 2021 01 14.
Article em En | MEDLINE | ID: mdl-33399453

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Ácidos Fosforosos / 5'-Nucleotidase Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Ácidos Fosforosos / 5'-Nucleotidase Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos