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Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase.
Brahmaiah, Dabbugoddu; Kanaka Durga Bhavani, Anagani; Aparna, Pasula; Sampath Kumar, Nangunoori; Solhi, Hélène; Le Guevel, Rémy; Baratte, Blandine; Ruchaud, Sandrine; Bach, Stéphane; Singh Jadav, Surender; Raji Reddy, Chada; Roisnel, Thierry; Mosset, Paul; Levoin, Nicolas; Grée, René.
Afiliação
  • Brahmaiah D; Chemveda Life Sciences India Pvt. Ltd., #B-11/1, IDA Uppal, Hyderabad 500039, Telangana, India; Jawaharlal Nehru Technological University Hyderabad, Kukatpally, Hyderabad 500 085, Telangana, India.
  • Kanaka Durga Bhavani A; Department of Chemistry, Osmania University, Hyderabad 500007, Telangana, India.
  • Aparna P; Jawaharlal Nehru Technological University Hyderabad, Kukatpally, Hyderabad 500 085, Telangana, India.
  • Sampath Kumar N; Chemveda Life Sciences India Pvt. Ltd., #B-11/1, IDA Uppal, Hyderabad 500039, Telangana, India.
  • Solhi H; Univ Rennes, Plateform ImPACcell, BIOSIT, F-35000 Rennes, France.
  • Le Guevel R; Univ Rennes, Plateform ImPACcell, BIOSIT, F-35000 Rennes, France.
  • Baratte B; Sorbonne Université, CNRS, FR 2424, Plateforme de criblage KISSf (Kinase Inhibitor Specialized Screening Facility), Station Biologique de Roscoff, CS 90074, 29688 Roscoff Cedex, France; Sorbonne Université, CNRS, UMR 8227, Integrative Biology of Marine Models Laboratory (LBI2M), Station Biologique d
  • Ruchaud S; Sorbonne Université, CNRS, UMR 8227, Integrative Biology of Marine Models Laboratory (LBI2M), Station Biologique de Roscoff, CS 90074, 29688 Roscoff Cedex, France.
  • Bach S; Sorbonne Université, CNRS, FR 2424, Plateforme de criblage KISSf (Kinase Inhibitor Specialized Screening Facility), Station Biologique de Roscoff, CS 90074, 29688 Roscoff Cedex, France; Sorbonne Université, CNRS, UMR 8227, Integrative Biology of Marine Models Laboratory (LBI2M), Station Biologique d
  • Singh Jadav S; CSIR-Indian Institute of Chemical Technology, Uppal Road, Tarnaka, Hyderabad 500007, TS, India.
  • Raji Reddy C; CSIR-Indian Institute of Chemical Technology, Uppal Road, Tarnaka, Hyderabad 500007, TS, India.
  • Roisnel T; Univ Rennes, CNRS, ISCR (Institut des Sciences Chimiques de Rennes), UMR 6226, F-35000 Rennes, France.
  • Mosset P; Univ Rennes, CNRS, ISCR (Institut des Sciences Chimiques de Rennes), UMR 6226, F-35000 Rennes, France.
  • Levoin N; Bioprojet-Biotech, 4 rue du Chesnay Beauregard, BP 96205, 35762 Saint Grégoire, France.
  • Grée R; Univ Rennes, CNRS, ISCR (Institut des Sciences Chimiques de Rennes), UMR 6226, F-35000 Rennes, France. Electronic address: rene.gree@univ-rennes1.fr.
Bioorg Med Chem ; 31: 115962, 2021 02 01.
Article em En | MEDLINE | ID: mdl-33422908
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Texto completo: 1 Base de dados: MEDLINE Assunto principal: Proteínas Tirosina Quinases / Proteínas Serina-Treonina Quinases / Inibidores de Proteínas Quinases / Descoberta de Drogas / Antineoplásicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Índia
Texto completo
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Texto completo: 1 Base de dados: MEDLINE Assunto principal: Proteínas Tirosina Quinases / Proteínas Serina-Treonina Quinases / Inibidores de Proteínas Quinases / Descoberta de Drogas / Antineoplásicos Limite: Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Índia