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A New Inhibitor of ADAM17 Composed of a Zinc-Binding Dithiol Moiety and a Specificity Pocket-Binding Appendage.
Tateishi, Hiroshi; Tateishi, Mika; Radwan, Mohamed O; Masunaga, Takuya; Kawatashiro, Kosuke; Oba, Yasunori; Oyama, Misato; Inoue-Kitahashi, Natsuki; Fujita, Mikako; Okamoto, Yoshinari; Otsuka, Masami.
Afiliação
  • Tateishi H; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Tateishi M; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Radwan MO; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Masunaga T; Chemistry of Natural Compounds Department, Pharmaceutical and Drug Industries Research Division, National Research Centre.
  • Kawatashiro K; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Oba Y; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Oyama M; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Inoue-Kitahashi N; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Fujita M; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Okamoto Y; Medicinal and Biological Chemistry Science Farm Joint Research Laboratory, Faculty of Life Sciences, Kumamoto University.
  • Otsuka M; Department of Instrumental Analysis, Faculty of Life Sciences, Kumamoto University.
Chem Pharm Bull (Tokyo) ; 69(11): 1123-1130, 2021.
Article em En | MEDLINE | ID: mdl-34719595

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Sulfonamidas / Tolueno / Proteína ADAM17 Limite: Humans Idioma: En Revista: Chem Pharm Bull (Tokyo) Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Sulfonamidas / Tolueno / Proteína ADAM17 Limite: Humans Idioma: En Revista: Chem Pharm Bull (Tokyo) Ano de publicação: 2021 Tipo de documento: Article