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Design, synthesis and molecular docking of new fused 1H-pyrroles, pyrrolo[3,2-d]pyrimidines and pyrrolo[3,2-e][1, 4]diazepine derivatives as potent EGFR/CDK2 inhibitors.
Belal, Amany; Abdel Gawad, Nagwa M; Mehany, Ahmed B M; Abourehab, Mohammed A S; Elkady, Hazem; Al-Karmalawy, Ahmed A; Ismael, Ahmed S.
Afiliação
  • Belal A; Medicinal Chemistry Department, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, Egypt.
  • Abdel Gawad NM; Department of Pharmaceutical Chemistry, College of Pharmacy, Taif University, Taif, Saudi Arabia.
  • Mehany ABM; Medicinal Chemistry Department, Faculty of Pharmacy, Cairo University, Giza, Egypt.
  • Abourehab MAS; Department of Zoology, Faculty of Science, Al-Azhar University, Nasr City, Egypt.
  • Elkady H; Department of Pharmaceutics, Faculty of Pharmacy, Umm Al-Qura University, Makkah, Saudi Arabia.
  • Al-Karmalawy AA; Department of Pharmaceutics and Industrial Pharmacy, College of Pharmacy, Minia University, Minia, Egypt.
  • Ismael AS; Pharmaceutical Medicinal Chemistry & Drug Design Department, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo, Egypt.
J Enzyme Inhib Med Chem ; 37(1): 1884-1902, 2022 Dec.
Article em En | MEDLINE | ID: mdl-35801486

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirimidinas / Antineoplásicos Limite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Egito

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirimidinas / Antineoplásicos Limite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Egito