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Bioisosteric Design Identifies Inhibitors of Mycobacterium tuberculosis DNA Gyrase ATPase Activity.
Kamsri, Bundit; Pakamwong, Bongkochawan; Thongdee, Paptawan; Phusi, Naruedon; Kamsri, Pharit; Punkvang, Auradee; Ketrat, Sombat; Saparpakorn, Patchreenart; Hannongbua, Supa; Sangswan, Jidapa; Suttisintong, Khomson; Sureram, Sanya; Kittakoop, Prasat; Hongmanee, Poonpilas; Santanirand, Pitak; Leanpolchareanchai, Jiraporn; Goudar, Kirsty E; Spencer, James; Mulholland, Adrian J; Pungpo, Pornpan.
Afiliação
  • Kamsri B; Department of Chemistry, Faculty of Science, Ubon Ratchathani University, Ubon Ratchathani 34190, Thailand.
  • Pakamwong B; Department of Chemistry, Faculty of Science, Ubon Ratchathani University, Ubon Ratchathani 34190, Thailand.
  • Thongdee P; Department of Chemistry, Faculty of Science, Ubon Ratchathani University, Ubon Ratchathani 34190, Thailand.
  • Phusi N; Department of Chemistry, Faculty of Science, Ubon Ratchathani University, Ubon Ratchathani 34190, Thailand.
  • Kamsri P; Division of Chemistry, Faculty of Science, Nakhon Phanom University, Nakhon Phanom 48000, Thailand.
  • Punkvang A; Division of Chemistry, Faculty of Science, Nakhon Phanom University, Nakhon Phanom 48000, Thailand.
  • Ketrat S; School of Information Science and Technology, Vidyasirimedhi Institute of Science and Technology, Rayong 21210, Thailand.
  • Saparpakorn P; Department of Chemistry, Faculty of Science, Kasetsart University, Bangkok 10900, Thailand.
  • Hannongbua S; Department of Chemistry, Faculty of Science, Kasetsart University, Bangkok 10900, Thailand.
  • Sangswan J; Department of Biological Science, Faculty of Science, Ubon Ratchathani University, Ubon Ratchathani 34190, Thailand.
  • Suttisintong K; National Nanotechnology Center, NSTDA, 111 Thailand Science Park, Klong Luang, Pathum Thani 12120, Thailand.
  • Sureram S; Chulabhorn Research Institute, Bangkok 10210, Thailand.
  • Kittakoop P; Chulabhorn Research Institute, Bangkok 10210, Thailand.
  • Hongmanee P; Chulabhorn Graduate Institute, Chemical Biology Program, Chulabhorn Royal Academy, Bangkok 10210, Thailand.
  • Santanirand P; Center of Excellence on Environmental Health and Toxicology (EHT), OPS, Ministry of Higher Education, Science, Research and Innovation, Bangkok 10210, Thailand.
  • Leanpolchareanchai J; Division of Microbiology, Department of Pathology, Faculty of Medicine, Ramathibodi Hospital, Mahidol University, Bangkok 10400, Thailand.
  • Goudar KE; Division of Microbiology, Department of Pathology, Faculty of Medicine, Ramathibodi Hospital, Mahidol University, Bangkok 10400, Thailand.
  • Spencer J; Department of Pharmacy, Faculty of Pharmacy, Mahidol University, 447 Sri-Ayuthaya Road,Rajathevi, Bangkok 10400, Thailand.
  • Mulholland AJ; School of Cellular and Molecular Medicine, Biomedical Sciences Building, University of Bristol, Bristol BS8 1TD, United Kingdom.
  • Pungpo P; School of Cellular and Molecular Medicine, Biomedical Sciences Building, University of Bristol, Bristol BS8 1TD, United Kingdom.
J Chem Inf Model ; 63(9): 2707-2718, 2023 05 08.
Article em En | MEDLINE | ID: mdl-37074047

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tuberculose / Mycobacterium tuberculosis Limite: Humans Idioma: En Revista: J Chem Inf Model Assunto da revista: INFORMATICA MEDICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Tailândia

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tuberculose / Mycobacterium tuberculosis Limite: Humans Idioma: En Revista: J Chem Inf Model Assunto da revista: INFORMATICA MEDICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Tailândia