Detalhe da pesquisa
1.
Versatile Click Linker Enabling Native Peptide Release from Nanocarriers upon Redox Trigger.
Bioconjug Chem
; 34(12): 2375-2386, 2023 12 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-38079189
2.
A New Class of Tunable Acid-Sensitive Linkers for Native Drug Release Based on the Trityl Protecting Group.
Bioconjug Chem
; 33(9): 1707-1715, 2022 Sep 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-35979909
3.
Synthesis of a tricyclic hexapeptide -via two consecutive ruthenium-catalyzed macrocyclization steps- with a constrained topology to mimic vancomycin's binding properties toward D-Ala-D-Ala dipeptide.
Bioorg Med Chem Lett
; 73: 128887, 2022 10 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-35835378
4.
Improving the aqueous solubility of HCV-E2 glycoprotein epitope mimics by cyclization using POLAR hinges.
J Pept Sci
; 26(1): e3222, 2020 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-31984607
5.
Design, Synthesis, and Evaluation of a Diazirine Photoaffinity Probe for Ligand-Based Receptor Capture Targeting G Protein-Coupled Receptors.
Mol Pharmacol
; 95(2): 196-209, 2019 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-30514721
6.
Molecular Construction of Sulfonamide Antisense Oligonucleotides.
J Org Chem
; 84(17): 10635-10648, 2019 09 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-31379169
7.
Immobilization by Surface Conjugation of Cyclic Peptides for Effective Mimicry of the HCV-Envelope E2 Protein as a Strategy toward Synthetic Vaccines.
Bioconjug Chem
; 29(4): 1091-1101, 2018 04 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-29382188
8.
Synthetic antibody protein mimics of infliximab by molecular scaffolding on novel CycloTriVeratrilene (CTV) derivatives.
Org Biomol Chem
; 16(29): 5254-5274, 2018 07 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-29892733
9.
Polar Hinges as Functionalized Conformational Constraints in (Bi)cyclic Peptides.
Chembiochem
; 18(4): 387-395, 2017 02 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-27982494
10.
An orthogonally protected CycloTriVeratrylene (CTV) as a highly pre-organized molecular scaffold for subsequent ligation of different cyclic peptides towards protein mimics.
Bioorg Med Chem
; 25(18): 5008-5015, 2017 09 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-28583807
11.
Potential peptidic proteasome inhibitors by incorporation of an electrophilic trap based on amino acid derived α-substituted sulfonyl fluorides.
Bioorg Med Chem
; 25(19): 5055-5063, 2017 10 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28734665
12.
Proteasome inhibition by new dual warhead containing peptido vinyl sulfonyl fluorides.
Bioorg Med Chem
; 24(16): 3429-35, 2016 08 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27316540
13.
Activity-based probes for rhomboid proteases discovered in a mass spectrometry-based assay.
Proc Natl Acad Sci U S A
; 110(7): 2472-7, 2013 Feb 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-23359682
14.
Synthesis of pyrazole containing α-amino acids via a highly regioselective condensation/aza-Michael reaction of ß-aryl α,ß-unsaturated ketones.
Org Biomol Chem
; 13(15): 4514-23, 2015 Apr 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-25774874
15.
Synthesis of nisin AB dicarba analogs using ring-closing metathesis: influence of sp(3) versus sp(2) hybridization of the α-carbon atom of residues dehydrobutyrine-2 and dehydroalanine-5 on the lipid II binding affinity.
Org Biomol Chem
; 13(21): 5997-6009, 2015 Jun 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-25940216
16.
Unusual binding of Grb2 protein to a bivalent polyproline-ligand immobilized on a SPR sensor: intermolecular bivalent binding.
Biochim Biophys Acta
; 1834(2): 524-35, 2013 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-23159538
17.
New properties of wheat bran: anti-biofilm activity and interference with bacteria quorum-sensing systems.
Environ Microbiol
; 16(5): 1346-53, 2014 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-24588934
18.
A versatile spectrophotometric protein tyrosine phosphatase assay based on 3-nitrophosphotyrosine containing substrates.
Anal Biochem
; 448: 9-13, 2014 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24309020
19.
Characterization and activity of an immobilized antimicrobial peptide containing bactericidal PEG-hydrogel.
Biomacromolecules
; 15(9): 3390-5, 2014 Sep 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-25109707
20.
Azide-alkyne cycloaddition affording enzymatically tunable bisubstrate based inhibitors of histone acetyltransferase PCAF.
Bioorg Med Chem Lett
; 24(1): 113-6, 2014 Jan 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-24345448