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Design, synthesis and pharmacological evaluation of novel polycyclic heteroarene ethers as PDE10A inhibitors: part II.
Das, Sanjib; Shelke, Dnyaneshwar E; Harde, Rajendra L; Avhad, Vijayshree B; Khairatkar-Joshi, Neelima; Gullapalli, Srinivas; Gupta, Praveen K; Gandhi, Maulik N; Bhateja, Deepak K; Bajpai, Malini; Joshi, Ashwini A; Marathe, Megha Y; Gudi, Girish S; Jadhav, Satyawan B; Mahat, Mahamad Yunnus A; Thomas, Abraham.
Afiliação
  • Das S; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Shelke DE; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Harde RL; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Avhad VB; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Khairatkar-Joshi N; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Gullapalli S; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Gupta PK; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Gandhi MN; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Bhateja DK; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Bajpai M; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Joshi AA; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Marathe MY; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Gudi GS; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Jadhav SB; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Mahat MY; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India.
  • Thomas A; Glenmark Research Centre, Glenmark Pharmaceuticals Ltd, MIDC, Mahape, Navi Mumbai 400 709, India. Electronic address: abraham_thomas@glenmarkpharma.com.
Bioorg Med Chem Lett ; 24(15): 3238-42, 2014 Aug 01.
Article em En | MEDLINE | ID: mdl-24980052

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Fosfodiesterase / Pirazinas / Piridinas / Desenho de Fármacos / Diester Fosfórico Hidrolases / Éteres Limite: Animals / Humans / Male Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Fosfodiesterase / Pirazinas / Piridinas / Desenho de Fármacos / Diester Fosfórico Hidrolases / Éteres Limite: Animals / Humans / Male Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Índia