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Synthesis and biological evaluation of some novel triazole hybrids of curcumin mimics and their selective anticancer activity against breast and prostate cancer cell lines.
Mandalapu, Dhanaraju; Saini, Karan S; Gupta, Sonal; Sharma, Vikas; Yaseen Malik, Mohd; Chaturvedi, Swati; Bala, Veenu; Thakur, Subhadra; Maikhuri, Jagdamba P; Wahajuddin, Muhammad; Konwar, Rituraj; Gupta, Gopal; Sharma, Vishnu Lal.
Afiliação
  • Mandalapu D; Medicinal & Process Chemistry Division, CSIR-Central Drug Research Institute, Sector 10, Jankipuram ext., Sitapur Road, Lucknow, Uttar Pradesh 226031, India.
  • Saini KS; Endocrinology Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Gupta S; Medicinal & Process Chemistry Division, CSIR-Central Drug Research Institute, Sector 10, Jankipuram ext., Sitapur Road, Lucknow, Uttar Pradesh 226031, India; Academy of Scientific and Innovative Research (AcSIR), New Delhi 110001, India.
  • Sharma V; Endocrinology Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Yaseen Malik M; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Chaturvedi S; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Bala V; Medicinal & Process Chemistry Division, CSIR-Central Drug Research Institute, Sector 10, Jankipuram ext., Sitapur Road, Lucknow, Uttar Pradesh 226031, India; Academy of Scientific and Innovative Research (AcSIR), New Delhi 110001, India.
  • Hamidullah; Endocrinology Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Thakur S; Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Raebareli 229010, India.
  • Maikhuri JP; Endocrinology Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Wahajuddin M; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Konwar R; Endocrinology Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Gupta G; Endocrinology Division, CSIR-Central Drug Research Institute, Sitapur Road, Lucknow 226031, India.
  • Sharma VL; Medicinal & Process Chemistry Division, CSIR-Central Drug Research Institute, Sector 10, Jankipuram ext., Sitapur Road, Lucknow, Uttar Pradesh 226031, India; Academy of Scientific and Innovative Research (AcSIR), New Delhi 110001, India. Electronic address: vl_sharma@cdri.res.in.
Bioorg Med Chem Lett ; 26(17): 4223-32, 2016 09 01.
Article em En | MEDLINE | ID: mdl-27496212

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Triazóis / Curcumina / Antineoplásicos Limite: Female / Humans / Male Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Triazóis / Curcumina / Antineoplásicos Limite: Female / Humans / Male Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Índia