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The new small tyrosine kinase inhibitor ARQ531 targets acute myeloid leukemia cells by disrupting multiple tumor-addicted programs.
Soncini, Debora; Orecchioni, Stefania; Ruberti, Samantha; Minetto, Paola; Martinuzzi, Claudia; Agnelli, Luca; Todoerti, Katia; Cagnetta, Antonia; Miglino, Maurizio; Clavio, Marino; Contini, Paola; Varaldo, Riccardo; Bergamaschi, Micaela; Guolo, Fabio; Passalacqua, Mario; Nencioni, Alessio; Monacelli, Fiammetta; Gobbi, Marco; Neri, Antonino; Abbadessa, Giovanni; Eathiraj, Sudharshan; Schwartz, Brian; Bertolini, Francesco; Lemoli, Roberto M; Cea, Michele.
Afiliação
  • Soncini D; University of Genoa, DiMI, Italy.
  • Orecchioni S; Laboratory of Hematology-Oncology European Institute of Oncology IRCCS, Milan, Italy.
  • Ruberti S; University of Genoa, DiMI, Italy.
  • Minetto P; University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
  • Martinuzzi C; University of Genoa, DiMI, Italy.
  • Agnelli L; Department of Oncology and Hemato-Oncology, University of Milan, Milan, Italy.
  • Todoerti K; Department of Oncology and Hemato-Oncology, University of Milan, Milan, Italy.
  • Cagnetta A; University of Genoa,University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
  • Miglino M; University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
  • Clavio M; University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
  • Contini P; University of Genoa, Department of Internal Medicine and Specialities (DiMI), Italy.
  • Varaldo R; Ospedale Policlinico San Martino, Genoa, Italy.
  • Bergamaschi M; University of Genoa, DiMI, Italy.
  • Guolo F; University of Genoa, DiMI, Italy.
  • Passalacqua M; University of Genoa, Department of Experimental Medicine (DIMES), Italy.
  • Nencioni A; University of Genoa, Department of Internal Medicine and Specialities (DiMI), Italy.
  • Monacelli F; University of Genoa, Department of Internal Medicine and Specialities (DiMI), Italy.
  • Gobbi M; University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
  • Neri A; Department of Oncology and Hemato-Oncology, University of Milan, Milan, Italy.
  • Abbadessa G; ArQule, One Wall Street, Burlington, MA, USA.
  • Eathiraj S; ArQule, One Wall Street, Burlington, MA, USA.
  • Schwartz B; ArQule, One Wall Street, Burlington, MA, USA.
  • Bertolini F; Laboratory of Hematology-Oncology European Institute of Oncology IRCCS, Milan, Italy.
  • Lemoli RM; University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
  • Cea M; University of Genoa, DiMI; IRCCS Ospedale Policlinico San Martino, Genoa, Italy.
Haematologica ; 105(10): 2420-2431, 2020 10 01.
Article em En | MEDLINE | ID: mdl-33054082

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Leucemia Mieloide Aguda / Inibidores de Proteínas Quinases Limite: Humans Idioma: En Revista: Haematologica Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Itália

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Leucemia Mieloide Aguda / Inibidores de Proteínas Quinases Limite: Humans Idioma: En Revista: Haematologica Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Itália