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Polycomb Paralog Chromodomain Inhibitors Active against Both CBX6 and CBX8*.
Milosevich, Natalia; Wilson, Chelsea R; Brown, Tyler M; Alpsoy, Aktan; Wang, Sijie; Connelly, Katelyn E; Sinclair, Kirsten A D; Ponio, Felino R; Hof, Rebecca; Dykhuizen, Emily C; Hof, Fraser.
Afiliação
  • Milosevich N; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
  • Wilson CR; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
  • Brown TM; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
  • Alpsoy A; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University and Purdue University Center for Cancer Research, 575 Stadium Mall Drive, West Lafayette, IN, 47906, USA.
  • Wang S; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University and Purdue University Center for Cancer Research, 575 Stadium Mall Drive, West Lafayette, IN, 47906, USA.
  • Connelly KE; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University and Purdue University Center for Cancer Research, 575 Stadium Mall Drive, West Lafayette, IN, 47906, USA.
  • Sinclair KAD; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
  • Ponio FR; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
  • Hof R; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
  • Dykhuizen EC; Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University and Purdue University Center for Cancer Research, 575 Stadium Mall Drive, West Lafayette, IN, 47906, USA.
  • Hof F; Department of Chemistry, University of Victoria, Victoria, BC, V8W 3V6, Canada.
ChemMedChem ; 16(19): 3027-3034, 2021 10 06.
Article em En | MEDLINE | ID: mdl-34174168

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Peptídeos / Proteínas do Grupo Polycomb / Complexo Repressor Polycomb 1 / Antineoplásicos Limite: Humans Idioma: En Revista: ChemMedChem Assunto da revista: FARMACOLOGIA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Canadá

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Peptídeos / Proteínas do Grupo Polycomb / Complexo Repressor Polycomb 1 / Antineoplásicos Limite: Humans Idioma: En Revista: ChemMedChem Assunto da revista: FARMACOLOGIA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Canadá