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Pentafluorosulfanyl (SF5) as a Superior 19F Magnetic Resonance Reporter Group: Signal Detection and Biological Activity of Teriflunomide Derivatives.
Prinz, Christian; Starke, Ludger; Ramspoth, Tizian-Frank; Kerkering, Janis; Martos Riaño, Vera; Paul, Jérôme; Neuenschwander, Martin; Oder, Andreas; Radetzki, Silke; Adelhoefer, Siegfried; Ramos Delgado, Paula; Aravina, Mariya; Millward, Jason M; Fillmer, Ariane; Paul, Friedemann; Siffrin, Volker; von Kries, Jens-Peter; Niendorf, Thoralf; Nazaré, Marc; Waiczies, Sonia.
Afiliação
  • Prinz C; Berlin Ultrahigh Field Facility (B.U.F.F.), Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Starke L; Experimental and Clinical Research Center, a joint cooperation between the Charité - Universitätsmedizin Berlin and the Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Ramspoth TF; Berlin Ultrahigh Field Facility (B.U.F.F.), Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Kerkering J; Medicinal Chemistry, Leibniz-Institut für Molekulare Pharmakologie (FMP), Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Martos Riaño V; Experimental and Clinical Research Center, a joint cooperation between the Charité - Universitätsmedizin Berlin and the Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Paul J; Medicinal Chemistry, Leibniz-Institut für Molekulare Pharmakologie (FMP), Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Neuenschwander M; Medicinal Chemistry, Leibniz-Institut für Molekulare Pharmakologie (FMP), Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Oder A; Screening Unit, Leibniz-Institut für Molekulare Pharmakologie (FMP), Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Radetzki S; Screening Unit, Leibniz-Institut für Molekulare Pharmakologie (FMP), Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Adelhoefer S; Screening Unit, Leibniz-Institut für Molekulare Pharmakologie (FMP), Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Ramos Delgado P; Berlin Ultrahigh Field Facility (B.U.F.F.), Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Aravina M; Berlin Ultrahigh Field Facility (B.U.F.F.), Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Millward JM; Experimental and Clinical Research Center, a joint cooperation between the Charité - Universitätsmedizin Berlin and the Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Fillmer A; Berlin Ultrahigh Field Facility (B.U.F.F.), Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Paul F; Berlin Ultrahigh Field Facility (B.U.F.F.), Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Siffrin V; Experimental and Clinical Research Center, a joint cooperation between the Charité - Universitätsmedizin Berlin and the Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • von Kries JP; Physikalisch-Technische Bundesanstalt (PTB), Abbestraße 2-12, 10587 Berlin, Germany.
  • Niendorf T; Experimental and Clinical Research Center, a joint cooperation between the Charité - Universitätsmedizin Berlin and the Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
  • Nazaré M; Charité - Universitätsmedizin Berlin, corporate member of Freie Universität Berlin, Humboldt-Universität zu Berlin, and Berlin Institute of Health (BIH), Charitéplatz 1, 10117 Berlin, Germany.
  • Waiczies S; Experimental and Clinical Research Center, a joint cooperation between the Charité - Universitätsmedizin Berlin and the Max Delbrück Center for Molecular Medicine in the Helmholtz Association, Robert Rössle Straße 10, 13125 Berlin, Germany.
ACS Sens ; 6(11): 3948-3956, 2021 11 26.
Article em En | MEDLINE | ID: mdl-34666481

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Crotonatos / Di-Hidro-Orotato Desidrogenase Tipo de estudo: Diagnostic_studies Limite: Animals Idioma: En Revista: ACS Sens Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Crotonatos / Di-Hidro-Orotato Desidrogenase Tipo de estudo: Diagnostic_studies Limite: Animals Idioma: En Revista: ACS Sens Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Alemanha