1.
Bioorg Med Chem Lett
; 16(23): 6086-90, 2006 Dec 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-16987661
RESUMO
A series of potent steroidal glucocorticoid receptor antagonists has been discovered. After conjugation to cholic acid, the compounds retained an affinity for GR in vitro and had modest in vivo efficacy.