Design and pharmacology of N-[(3R)-1,2,3,4-tetrahydroisoquinolinium- 3-ylcarbonyl]-(1R)-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1H-1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine (1), a potent, selective, melanocortin subtype-4 receptor agonist.
J Med Chem
; 45(21): 4589-93, 2002 Oct 10.
Article
em En
| MEDLINE
| ID: mdl-12361385
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Base de dados:
MEDLINE
Assunto principal:
Triazóis
/
Receptores da Corticotropina
/
Tetra-Hidroisoquinolinas
/
Isoquinolinas
Idioma:
En
Ano de publicação:
2002
Tipo de documento:
Article