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In vitro and in vivo comparison of two non-peptide tachykinin NK3 receptor antagonists: Improvements in efficacy achieved through enhanced brain penetration or altered pharmacological characteristics.
Dawson, Lee A; Langmead, Christopher J; Dada, Adeshola; Watson, Jeannette M; Wu, Zining; de la Flor, Raúl; Jones, Gareth A; Cluderay, Jane E; Southam, Eric; Murkitt, Graham S; Hill, Mark D; Jones, Declan N C; Davies, Ceri H; Hagan, Jim J; Smith, Paul W.
Afiliação
  • Dawson LA; Neurosciences Centre of Excellence for Drug Discovery, GlaxoSmithKline, New Frontiers Science Park, Harlow, Essex, UK. Lee_Dawson@eisai.net
Eur J Pharmacol ; 627(1-3): 106-14, 2010 Feb 10.
Article em En | MEDLINE | ID: mdl-19879867

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinolinas / Encéfalo / Receptores de Taquicininas / Aminoquinolinas Idioma: En Ano de publicação: 2010 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinolinas / Encéfalo / Receptores de Taquicininas / Aminoquinolinas Idioma: En Ano de publicação: 2010 Tipo de documento: Article