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Identification of Potent and Selective Inhibitors of the Plasmodium falciparum M18 Aspartyl Aminopeptidase (PfM18AAP) of Human Malaria via High-Throughput Screening.
Spicer, Timothy; Fernandez-Vega, Virneliz; Chase, Peter; Scampavia, Louis; To, Joyce; Dalton, John P; Da Silva, Fabio L; Skinner-Adams, Tina S; Gardiner, Donald L; Trenholme, Katharine R; Brown, Christopher L; Ghosh, Partha; Porubsky, Patrick; Wang, Jenna L; Whipple, David A; Schoenen, Frank J; Hodder, Peter.
Afiliação
  • Spicer T; The Scripps Research Institute Molecular Screening Center, Scripps Florida, Jupiter, FL, USA.
  • Fernandez-Vega V; The Scripps Research Institute Molecular Screening Center, Scripps Florida, Jupiter, FL, USA.
  • Chase P; The Scripps Research Institute Molecular Screening Center, Scripps Florida, Jupiter, FL, USA.
  • Scampavia L; The Scripps Research Institute Molecular Screening Center, Scripps Florida, Jupiter, FL, USA.
  • To J; Institute for Biotechnology of Infectious Diseases, University of Technology Sydney, Sydney, Australia.
  • Dalton JP; Institute for Biotechnology of Infectious Diseases, University of Technology Sydney, Sydney, Australia Institute of Parasitology, McGill University, Quebec, Canada.
  • Da Silva FL; Malaria Biology Laboratory, The Queensland Institute of Medical Research, Brisbane, Australia.
  • Skinner-Adams TS; Malaria Biology Laboratory, The Queensland Institute of Medical Research, Brisbane, Australia.
  • Gardiner DL; Malaria Biology Laboratory, The Queensland Institute of Medical Research, Brisbane, Australia.
  • Trenholme KR; Malaria Biology Laboratory, The Queensland Institute of Medical Research, Brisbane, Australia.
  • Brown CL; School of Biomolecular and Physical Sciences, Griffith University, Brisbane, Australia.
  • Ghosh P; The University of Kansas Specialized Chemistry Center, Lawrence, KS, USA.
  • Porubsky P; The University of Kansas Specialized Chemistry Center, Lawrence, KS, USA.
  • Wang JL; The University of Kansas Specialized Chemistry Center, Lawrence, KS, USA.
  • Whipple DA; The University of Kansas Specialized Chemistry Center, Lawrence, KS, USA.
  • Schoenen FJ; The University of Kansas Specialized Chemistry Center, Lawrence, KS, USA.
  • Hodder P; The Scripps Research Institute Molecular Screening Center, Scripps Florida, Jupiter, FL, USA hodderp@scripps.edu.
J Biomol Screen ; 19(7): 1107-15, 2014 Aug.
Article em En | MEDLINE | ID: mdl-24619116

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Malária Falciparum / Glutamil Aminopeptidase / Aminopeptidases / Antimaláricos Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Malária Falciparum / Glutamil Aminopeptidase / Aminopeptidases / Antimaláricos Idioma: En Ano de publicação: 2014 Tipo de documento: Article