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Synthesis and pharmacological evaluation of M4 muscarinic receptor positive allosteric modulators derived from VU10004.
Huynh, Tracey; Valant, Celine; Crosby, Ian T; Sexton, Patrick M; Christopoulos, Arthur; Capuano, Ben.
Afiliação
  • Huynh T; †Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia.
  • Valant C; †Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia.
  • Crosby IT; †Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia.
  • Sexton PM; †Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia.
  • Christopoulos A; †Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia.
  • Capuano B; †Medicinal Chemistry and ‡Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 381-399 Royal Parade, Parkville VIC 3052, Australia.
ACS Chem Neurosci ; 6(6): 838-44, 2015 Jun 17.
Article em En | MEDLINE | ID: mdl-25857219

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Agonistas Colinérgicos / Receptor Muscarínico M4 / Tienopiridinas Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Agonistas Colinérgicos / Receptor Muscarínico M4 / Tienopiridinas Idioma: En Ano de publicação: 2015 Tipo de documento: Article