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SAR Studies of Exosite-Binding Substrate-Selective Inhibitors of A Disintegrin And Metalloprotease 17 (ADAM17) and Application as Selective in Vitro Probes.
Knapinska, Anna M; Dreymuller, Daniela; Ludwig, Andreas; Smith, Lyndsay; Golubkov, Vladislav; Sohail, Anjum; Fridman, Rafael; Giulianotti, Marc; LaVoi, Travis M; Houghten, Richard A; Fields, Gregg B; Minond, Dmitriy.
Afiliação
  • Knapinska AM; ∥Florida Atlantic University, 5353 Parkside Drive, Jupiter, Florida 33458, United States.
  • Dreymuller D; ⊥Institute of Pharmacology and Toxicology, RWTH Aachen University, Wendlingweg 2, 52074 Aachen, Germany.
  • Ludwig A; ⊥Institute of Pharmacology and Toxicology, RWTH Aachen University, Wendlingweg 2, 52074 Aachen, Germany.
  • Smith L; ∥Florida Atlantic University, 5353 Parkside Drive, Jupiter, Florida 33458, United States.
  • Golubkov V; ‡Sanford-Burnham Medical Research Institute, 10901 North Torrey Pines Road, La Jolla, California 92037, United States.
  • Sohail A; §Wayne State University, 8200 Scott Hall, 540 East Canfield Avenue, Detroit, Michigan 48201, United States.
  • Fridman R; §Wayne State University, 8200 Scott Hall, 540 East Canfield Avenue, Detroit, Michigan 48201, United States.
  • Giulianotti M; †Torrey Pines Institute for Molecular Studies, 11350 SW Village Parkway, Port St. Lucie, Florida 34987, United States.
  • LaVoi TM; ∇Department of Chemistry, Center for Drug Discovery and Innovation, University of South Florida, Tampa, Florida 33612, United States.
  • Houghten RA; †Torrey Pines Institute for Molecular Studies, 11350 SW Village Parkway, Port St. Lucie, Florida 34987, United States.
  • Fields GB; †Torrey Pines Institute for Molecular Studies, 11350 SW Village Parkway, Port St. Lucie, Florida 34987, United States.
  • Minond D; ∥Florida Atlantic University, 5353 Parkside Drive, Jupiter, Florida 33458, United States.
J Med Chem ; 58(15): 5808-24, 2015 Aug 13.
Article em En | MEDLINE | ID: mdl-26192023

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sondas Moleculares / Proteínas ADAM Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sondas Moleculares / Proteínas ADAM Idioma: En Ano de publicação: 2015 Tipo de documento: Article