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Potent and Selective Inhibitors of Histone Deacetylase-3 Containing Chiral Oxazoline Capping Groups and a N-(2-Aminophenyl)-benzamide Binding Unit.
Marson, Charles M; Matthews, Christopher J; Atkinson, Stephen J; Lamadema, Nermina; Thomas, N Shaun B.
Afiliação
  • Marson CM; Department of Chemistry, University College London , Christopher Ingold Laboratories, 20 Gordon Street, London WC1H OAJ, U.K.
  • Matthews CJ; Department of Chemistry, University College London , Christopher Ingold Laboratories, 20 Gordon Street, London WC1H OAJ, U.K.
  • Atkinson SJ; Epinova DPU, Immuno-Inflammation Therapy Area Unit, GlaxoSmithKline , Gunnels Wood Road, Stevenage, Herts SG1 2NY, U.K.
  • Lamadema N; Department of Haematological Medicine, Leukaemia Sciences Laboratories, Rayne Institute, King's College London , 123 Coldharbour Lane, London SE5 9NU, U.K.
  • Thomas NS; Department of Haematological Medicine, Leukaemia Sciences Laboratories, Rayne Institute, King's College London , 123 Coldharbour Lane, London SE5 9NU, U.K.
J Med Chem ; 58(17): 6803-18, 2015 Sep 10.
Article em En | MEDLINE | ID: mdl-26287310

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxazóis / Benzamidas / Inibidores de Histona Desacetilases / Histona Desacetilases / Anilidas Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxazóis / Benzamidas / Inibidores de Histona Desacetilases / Histona Desacetilases / Anilidas Idioma: En Ano de publicação: 2015 Tipo de documento: Article