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Novel Series of Dihydropyridinone P2X7 Receptor Antagonists.
Lopez-Tapia, Francisco; Walker, Keith A M; Brotherton-Pleiss, Christine; Caroon, Joanie; Nitzan, Dov; Lowrie, Lee; Gleason, Shelley; Zhao, Shu-Hai; Berger, Jacob; Cockayne, Debra; Phippard, Deborah; Suttmann, Rebecca; Fitch, William L; Bourdet, David; Rege, Pankaj; Huang, Xiaojun; Broadbent, Scott; Dvorak, Charles; Zhu, Jiang; Wagner, Paul; Padilla, Fernando; Loe, Brad; Jahangir, Alam; Alker, André.
Afiliação
  • Lopez-Tapia F; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Walker KA; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Brotherton-Pleiss C; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Caroon J; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Nitzan D; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Lowrie L; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Gleason S; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Zhao SH; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Berger J; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Cockayne D; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Phippard D; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Suttmann R; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Fitch WL; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Bourdet D; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Rege P; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Huang X; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Broadbent S; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Dvorak C; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Zhu J; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Wagner P; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Padilla F; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Loe B; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Jahangir A; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
  • Alker A; Hoffmann-La Roche, Inc. , 340 Kingsland Street, Nutley, New Jersey 07110, United States.
J Med Chem ; 58(21): 8413-26, 2015 Nov 12.
Article em En | MEDLINE | ID: mdl-26460788

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridonas / Receptores Purinérgicos P2X7 / Antagonistas do Receptor Purinérgico P2X Idioma: En Ano de publicação: 2015 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Piridonas / Receptores Purinérgicos P2X7 / Antagonistas do Receptor Purinérgico P2X Idioma: En Ano de publicação: 2015 Tipo de documento: Article