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Biased agonism: An emerging paradigm in GPCR drug discovery.
Rankovic, Zoran; Brust, Tarsis F; Bohn, Laura M.
Afiliação
  • Rankovic Z; Discovery Chemistry and Research Technologies, Eli Lilly and Company, 893 South Delaware Street, Indianapolis, IN 46285, USA. Electronic address: rankovic_zoran@lilly.com.
  • Brust TF; Department of Molecular Therapeutics, and Department of Neuroscience, The Scripps Research Institute, Jupiter, FL 33458, USA.
  • Bohn LM; Department of Molecular Therapeutics, and Department of Neuroscience, The Scripps Research Institute, Jupiter, FL 33458, USA. Electronic address: lbohn@scripps.edu.
Bioorg Med Chem Lett ; 26(2): 241-250, 2016 Jan 15.
Article em En | MEDLINE | ID: mdl-26707396

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Arrestinas / Receptores Acoplados a Proteínas G / Descoberta de Drogas Idioma: En Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Arrestinas / Receptores Acoplados a Proteínas G / Descoberta de Drogas Idioma: En Ano de publicação: 2016 Tipo de documento: Article