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Discovery of new [1,4]dioxino[2,3-f]quinazoline-based inhibitors of EGFR including the T790M/L858R mutant.
Qin, Xuemei; Li, Zhipeng; Yang, Leifu; Liu, Peng; Hu, Liming; Zeng, Chengchu; Pan, Zhiyong.
Afiliação
  • Qin X; College of Life Science and Bioengineering, Beijing University of Technology, Beijing 100124, China.
  • Li Z; College of Life Science and Bioengineering, Beijing University of Technology, Beijing 100124, China.
  • Yang L; Beijing Dalitai Pharmaceutical Technology Co., Ltd, Beijing 100176, China.
  • Liu P; Guangzhou Institute of Biomedicine and Health, Chinese Academy of Science, Guangzhou 510530, China.
  • Hu L; College of Life Science and Bioengineering, Beijing University of Technology, Beijing 100124, China. Electronic address: huliming@bjut.edu.cn.
  • Zeng C; College of Life Science and Bioengineering, Beijing University of Technology, Beijing 100124, China.
  • Pan Z; Beijing Dalitai Pharmaceutical Technology Co., Ltd, Beijing 100176, China.
Bioorg Med Chem ; 24(13): 2871-2881, 2016 07 01.
Article em En | MEDLINE | ID: mdl-27234887

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinazolinas / Receptores ErbB Idioma: En Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Quinazolinas / Receptores ErbB Idioma: En Ano de publicação: 2016 Tipo de documento: Article