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Loop-F of the α-subunit determines the pharmacologic profile of novel competitive inhibitors of GABAA receptors.
Mihalik, Balázs; Pálvölgyi, Adrienn; Bogár, Ferenc; Megyeri, Katalin; Ling, István; Barkóczy, József; Bartha, Ferenc; Martinek, Tamás A; Gacsályi, István; Antoni, Ferenc A.
Afiliação
  • Mihalik B; Division of Preclinical Research, Egis Pharmaceuticals PLC, Hungary.
  • Pálvölgyi A; Division of Preclinical Research, Egis Pharmaceuticals PLC, Hungary.
  • Bogár F; MTA-SZTE Supramolecular and Nanostructured Materials Research Group of HAS, University of Szeged, Hungary.
  • Megyeri K; Division of Preclinical Research, Egis Pharmaceuticals PLC, Hungary.
  • Ling I; Chemical Research Division, Egis Pharmaceuticals PLC, Budapest, Hungary.
  • Barkóczy J; Chemical Research Division, Egis Pharmaceuticals PLC, Budapest, Hungary.
  • Bartha F; Department of Medical Chemistry, University of Szeged, Hungary.
  • Martinek TA; Institute of Pharmaceutical Analysis, SZTE-MTA Lendület Foldamer Research Group, University of Szeged, Szeged, Hungary.
  • Gacsályi I; Division of Preclinical Research, Egis Pharmaceuticals PLC, Hungary.
  • Antoni FA; Division of Preclinical Research, Egis Pharmaceuticals PLC, Hungary. Electronic address: franzantoni@gmail.com.
Eur J Pharmacol ; 798: 129-136, 2017 Mar 05.
Article em En | MEDLINE | ID: mdl-28153485

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Benzodiazepinas / Receptores de GABA-A / Subunidades Proteicas / Antagonistas de Receptores de GABA-A Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Benzodiazepinas / Receptores de GABA-A / Subunidades Proteicas / Antagonistas de Receptores de GABA-A Idioma: En Ano de publicação: 2017 Tipo de documento: Article