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1,6-Cyclophellitol Cyclosulfates: A New Class of Irreversible Glycosidase Inhibitor.
Artola, Marta; Wu, Liang; Ferraz, Maria J; Kuo, Chi-Lin; Raich, Lluís; Breen, Imogen Z; Offen, Wendy A; Codée, Jeroen D C; van der Marel, Gijsbert A; Rovira, Carme; Aerts, Johannes M F G; Davies, Gideon J; Overkleeft, Herman S.
Afiliação
  • Artola M; Department of Bio-organic Synthesis and Department of Medical Biochemistry, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Wu L; Department of Chemistry, University of York, Heslington, York, YO10 5DD, U.K.
  • Ferraz MJ; Department of Bio-organic Synthesis and Department of Medical Biochemistry, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Kuo CL; Department of Bio-organic Synthesis and Department of Medical Biochemistry, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Raich L; Departament de Química Inorgànica i Orgànica (Secció de Química Orgànica) and Institut de Química Teòrica i Computacional (IQTCUB), Universitat de Barcelona, Martí i Franquès 1, 08028 Barcelona, Spain.
  • Breen IZ; Department of Chemistry, University of York, Heslington, York, YO10 5DD, U.K.
  • Offen WA; Department of Chemistry, University of York, Heslington, York, YO10 5DD, U.K.
  • Codée JDC; Department of Bio-organic Synthesis and Department of Medical Biochemistry, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • van der Marel GA; Department of Bio-organic Synthesis and Department of Medical Biochemistry, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Rovira C; Departament de Química Inorgànica i Orgànica (Secció de Química Orgànica) and Institut de Química Teòrica i Computacional (IQTCUB), Universitat de Barcelona, Martí i Franquès 1, 08028 Barcelona, Spain.
  • Aerts JMFG; Fundació Catalana de Recerca i Estudis Avançats (ICREA), Passeig Lluís Companys 23, 08010 Barcelona, Spain.
  • Davies GJ; Department of Bio-organic Synthesis and Department of Medical Biochemistry, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Overkleeft HS; Department of Chemistry, University of York, Heslington, York, YO10 5DD, U.K.
ACS Cent Sci ; 3(7): 784-793, 2017 Jul 26.
Article em En | MEDLINE | ID: mdl-28776021

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2017 Tipo de documento: Article