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Direct NMR Probing of Hydration Shells of Protein Ligand Interfaces and Its Application to Drug Design.
Geist, Leonhard; Mayer, Moriz; Cockcroft, Xiao-Ling; Wolkerstorfer, Bernhard; Kessler, Dirk; Engelhardt, Harald; McConnell, Darryl B; Konrat, Robert.
Afiliação
  • Geist L; Christian Doppler Laboratory for High-Content Structural Biology and Biotechnology, Department of Structural and Computational Biology, University of Vienna , Campus Vienna Biocenter 5, A-1030 Vienna, Austria.
  • Mayer M; Boehringer Ingelheim RCV GmbH & Co. KG , Dr.-Boehringer-Gasse 5-11, A-1121 Vienna, Austria.
  • Cockcroft XL; Boehringer Ingelheim RCV GmbH & Co. KG , Dr.-Boehringer-Gasse 5-11, A-1121 Vienna, Austria.
  • Wolkerstorfer B; Boehringer Ingelheim RCV GmbH & Co. KG , Dr.-Boehringer-Gasse 5-11, A-1121 Vienna, Austria.
  • Kessler D; Boehringer Ingelheim RCV GmbH & Co. KG , Dr.-Boehringer-Gasse 5-11, A-1121 Vienna, Austria.
  • Engelhardt H; Boehringer Ingelheim RCV GmbH & Co. KG , Dr.-Boehringer-Gasse 5-11, A-1121 Vienna, Austria.
  • McConnell DB; Boehringer Ingelheim RCV GmbH & Co. KG , Dr.-Boehringer-Gasse 5-11, A-1121 Vienna, Austria.
  • Konrat R; Christian Doppler Laboratory for High-Content Structural Biology and Biotechnology, Department of Structural and Computational Biology, University of Vienna , Campus Vienna Biocenter 5, A-1030 Vienna, Austria.
J Med Chem ; 60(21): 8708-8715, 2017 11 09.
Article em En | MEDLINE | ID: mdl-28910100

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Água / Desenho de Fármacos / Proteínas / Ressonância Magnética Nuclear Biomolecular Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Água / Desenho de Fármacos / Proteínas / Ressonância Magnética Nuclear Biomolecular Idioma: En Ano de publicação: 2017 Tipo de documento: Article