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G-Quadruplex Identification in the Genome of Protozoan Parasites Points to Naphthalene Diimide Ligands as New Antiparasitic Agents.
Belmonte-Reche, Efres; Martínez-García, Marta; Guédin, Aurore; Zuffo, Michela; Arévalo-Ruiz, Matilde; Doria, Filippo; Campos-Salinas, Jenny; Maynadier, Marjorie; López-Rubio, José Juan; Freccero, Mauro; Mergny, Jean-Louis; Pérez-Victoria, José María; Morales, Juan Carlos.
Afiliação
  • Belmonte-Reche E; Department of Biochemistry and Molecular Pharmacology, Instituto de Parasitología y Biomedicina, CSIC , PTS Granada, Avda. del Conocimiento, 17, 18016 Armilla, Granada, Spain.
  • Martínez-García M; Department of Biochemistry and Molecular Pharmacology, Instituto de Parasitología y Biomedicina, CSIC , PTS Granada, Avda. del Conocimiento, 17, 18016 Armilla, Granada, Spain.
  • Guédin A; ARNA Laboratory, Université de Bordeaux, Inserm U1212, CNRS UMR5320, Institut Européen de Chimie Biologie (IECB), 2 Rue Robert Escarpit, 33607 Pessac, France.
  • Zuffo M; Department of Chemistry, University of Pavia , Via Taramelli 10, 27100 Pavia, Italy.
  • Arévalo-Ruiz M; Department of Biochemistry and Molecular Pharmacology, Instituto de Parasitología y Biomedicina, CSIC , PTS Granada, Avda. del Conocimiento, 17, 18016 Armilla, Granada, Spain.
  • Doria F; Department of Chemistry, University of Pavia , Via Taramelli 10, 27100 Pavia, Italy.
  • Campos-Salinas J; Department of Biochemistry and Molecular Pharmacology, Instituto de Parasitología y Biomedicina, CSIC , PTS Granada, Avda. del Conocimiento, 17, 18016 Armilla, Granada, Spain.
  • Maynadier M; Dynamique des Interactions Membranaires Normales et Pathologiques, CNRS UMR 5235, Université de Montpellier, 34095 Montpellier, France.
  • López-Rubio JJ; CNRS, 5290, IRD 224, University of Montpellier (UMR "MiVEGEC"), INSERM, 34394 Montpellier, France.
  • Freccero M; Department of Chemistry, University of Pavia , Via Taramelli 10, 27100 Pavia, Italy.
  • Mergny JL; ARNA Laboratory, Université de Bordeaux, Inserm U1212, CNRS UMR5320, Institut Européen de Chimie Biologie (IECB), 2 Rue Robert Escarpit, 33607 Pessac, France.
  • Pérez-Victoria JM; Institute of Biophysics , AS CR, v.v.i. Kralovopolska 135, 612 65 Brno, Czech Republic.
  • Morales JC; Department of Biochemistry and Molecular Pharmacology, Instituto de Parasitología y Biomedicina, CSIC , PTS Granada, Avda. del Conocimiento, 17, 18016 Armilla, Granada, Spain.
J Med Chem ; 61(3): 1231-1240, 2018 02 08.
Article em En | MEDLINE | ID: mdl-29323491

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Genoma de Protozoário / Quadruplex G / Imidas / Naftalenos / Antiparasitários Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Genoma de Protozoário / Quadruplex G / Imidas / Naftalenos / Antiparasitários Idioma: En Ano de publicação: 2018 Tipo de documento: Article