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Pevonedistat, a first-in-class NEDD8-activating enzyme inhibitor, combined with azacitidine in patients with AML.
Swords, Ronan T; Coutre, Steven; Maris, Michael B; Zeidner, Joshua F; Foran, James M; Cruz, Jose; Erba, Harry P; Berdeja, Jesus G; Tam, Wayne; Vardhanabhuti, Saran; Pawlikowska-Dobler, Iwona; Faessel, Hélène M; Dash, Ajeeta B; Sedarati, Farhad; Dezube, Bruce J; Faller, Douglas V; Savona, Michael R.
Afiliação
  • Swords RT; Sylvester Comprehensive Cancer Center, University of Miami, Miami, FL.
  • Coutre S; Department of Medicine, Stanford University, Stanford, CA.
  • Maris MB; Colorado Blood Cancer Institute, Denver, CO.
  • Zeidner JF; Lineberger Comprehensive Cancer Center, University of North Carolina, Chapel Hill, NC.
  • Foran JM; Mayo Clinic Cancer Center, Jacksonville, FL.
  • Cruz J; Texas Transplant Institute, San Antonio, TX.
  • Erba HP; UAB Comprehensive Cancer Center, University of Alabama at Birmingham, Birmingham, AL.
  • Berdeja JG; Sarah Cannon Research Institute, Nashville, TN.
  • Tam W; Department of Pathology and Laboratory Medicine, Weill Cornell Medicine, New York, NY.
  • Vardhanabhuti S; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Pawlikowska-Dobler I; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Faessel HM; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Dash AB; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Sedarati F; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Dezube BJ; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Faller DV; Millennium Pharmaceuticals, Inc., Cambridge, MA; and.
  • Savona MR; Vanderbilt-Ingram Cancer Center, Vanderbilt University School of Medicine, Nashville, TN.
Blood ; 131(13): 1415-1424, 2018 03 29.
Article em En | MEDLINE | ID: mdl-29348128

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirimidinas / Azacitidina / Leucemia Mieloide Aguda / Ciclopentanos / Enzimas de Conjugação de Ubiquitina / Inibidores Enzimáticos / Proteínas de Neoplasias Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirimidinas / Azacitidina / Leucemia Mieloide Aguda / Ciclopentanos / Enzimas de Conjugação de Ubiquitina / Inibidores Enzimáticos / Proteínas de Neoplasias Idioma: En Ano de publicação: 2018 Tipo de documento: Article