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Discovery of a Potent Grp94 Selective Inhibitor with Anti-Inflammatory Efficacy in a Mouse Model of Ulcerative Colitis.
Jiang, Fen; Guo, An-Ping; Xu, Jia-Chen; You, Qi-Dong; Xu, Xiao-Li.
Afiliação
  • Jiang F; State Key Laboratory of Natural Medicines and Jiang Su Key Laboratory of Drug Design and Optimization , China Pharmaceutical University , Nanjing 210009 , China.
  • Guo AP; Department of Medicinal Chemistry, School of Pharmacy , China Pharmaceutical University , Nanjing 210009 , China.
  • Xu JC; State Key Laboratory of Natural Medicines and Jiang Su Key Laboratory of Drug Design and Optimization , China Pharmaceutical University , Nanjing 210009 , China.
  • You QD; Department of Medicinal Chemistry, School of Pharmacy , China Pharmaceutical University , Nanjing 210009 , China.
  • Xu XL; State Key Laboratory of Natural Medicines and Jiang Su Key Laboratory of Drug Design and Optimization , China Pharmaceutical University , Nanjing 210009 , China.
J Med Chem ; 61(21): 9513-9533, 2018 11 08.
Article em En | MEDLINE | ID: mdl-30351001

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Colite Ulcerativa / Proteínas de Choque Térmico HSP70 / Descoberta de Drogas / Proteínas de Membrana / Anti-Inflamatórios Idioma: En Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Colite Ulcerativa / Proteínas de Choque Térmico HSP70 / Descoberta de Drogas / Proteínas de Membrana / Anti-Inflamatórios Idioma: En Ano de publicação: 2018 Tipo de documento: Article