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Identification of N-Substituted Triazolo-azetidines as Novel Antibacterials using pDualrep2 HTS Platform.
Ivanenkov, Yan A; Yamidanov, Renat S; Osterman, Ilya A; Sergiev, Petr V; Aladinskiy, Vladimir A; Aladinskaya, Anastasia V; Terentiev, Victor A; Veselov, Mark S; Ayginin, Andrey A; Skvortsov, Dmitry A; Komarova, Katerina S; Chemeris, Alexey V; Baimiev, Alexey Kh; Sofronova, Alina A; Malyshev, Alexander S; Machulkin, Alexey E; Petrov, Rostislav A; Bezrukov, Dmitry S; Filkov, Gleb I; Puchinina, Maria M; Zainullina, Liana F; Maximova, Marina A; Zileeva, Zulfiya R; Vakhitova, Yulia V; Dontsova, Olga A.
Afiliação
  • Ivanenkov YA; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Yamidanov RS; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Osterman IA; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Sergiev PV; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Aladinskiy VA; ChemDiv, 6605 Nancy Ridge Drive, San Diego, CA 92121, United States.
  • Aladinskaya AV; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Terentiev VA; Lomonosov Moscow State University, Chemistry Dept, Leninskie gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.
  • Veselov MS; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Ayginin AA; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Skvortsov DA; Lomonosov Moscow State University, Department of Chemistry and A.N. Belozersky Institute of Physico-Chemical Biology, Moscow, Russian Federation.
  • Komarova KS; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Chemeris AV; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Baimiev AK; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Sofronova AA; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Malyshev AS; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Machulkin AE; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Petrov RA; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Bezrukov DS; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Filkov GI; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Puchinina MM; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Zainullina LF; Institute of Biochemistry and Genetics Russian Academy of Science (IBG RAS) Ufa Scientific Centre, Oktyabrya Prospekt 71, 450054, Ufa, Russian Federation.
  • Maximova MA; Moscow Institute of Physics and Technology (State University), 9 Institutskiy lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation.
  • Zileeva ZR; Lomonosov Moscow State University, Department of Chemistry and A.N. Belozersky Institute of Physico-Chemical Biology, Moscow, Russian Federation.
  • Vakhitova YV; Skolkovo Institute of Science and Technology, Skolkovo, Russian Federation.
  • Dontsova OA; Lomonosov Moscow State University, Department of Chemistry and A.N. Belozersky Institute of Physico-Chemical Biology, Moscow, Russian Federation.
Comb Chem High Throughput Screen ; 22(5): 346-354, 2019 08 08.
Article em En | MEDLINE | ID: mdl-30987560

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Azetidinas / Antibacterianos Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Azetidinas / Antibacterianos Idioma: En Ano de publicação: 2019 Tipo de documento: Article