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Identification and Characterization of Approved Drugs and Drug-Like Compounds as Covalent Escherichia coli ClpP Inhibitors.
Sassetti, Elisa; Durante Cruz, Cristina; Tammela, Päivi; Winterhalter, Mathias; Augustyns, Koen; Gribbon, Philip; Windshügel, Björn.
Afiliação
  • Sassetti E; Fraunhofer Institute for Molecular Biology and Applied Ecology IME, ScreeningPort, 22525 Hamburg, Germany. eli.sassetti@gmail.com.
  • Durante Cruz C; Drug Research Program, Division of Pharmaceutical Biosciences, University of Helsinki, FI-00014 Helsinki, Finland. eli.sassetti@gmail.com.
  • Tammela P; Drug Research Program, Division of Pharmaceutical Biosciences, University of Helsinki, FI-00014 Helsinki, Finland. cristina.durantecruz@helsinki.fi.
  • Winterhalter M; Drug Research Program, Division of Pharmaceutical Biosciences, University of Helsinki, FI-00014 Helsinki, Finland. paivi.tammela@helsinki.fi.
  • Augustyns K; Department of Life Sciences and Chemistry, Jacobs University Bremen gGmbH, 28759 Bremen, Germany. m.winterhalter@jacobs-university.de.
  • Gribbon P; Laboratory of Medicinal Chemistry, University of Antwerp, B-2610 Antwerp, Belgium. koen.augustyns@uantwerpen.be.
  • Windshügel B; Fraunhofer Institute for Molecular Biology and Applied Ecology IME, ScreeningPort, 22525 Hamburg, Germany. philip.gribbon@ime.fraunhofer.de.
Int J Mol Sci ; 20(11)2019 May 31.
Article em En | MEDLINE | ID: mdl-31159170

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Proteínas de Escherichia coli / Endopeptidase Clp / Descoberta de Drogas / Antibacterianos Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Proteínas de Escherichia coli / Endopeptidase Clp / Descoberta de Drogas / Antibacterianos Idioma: En Ano de publicação: 2019 Tipo de documento: Article