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Synthesis, Antimicrobial Activity and Molecular Docking of Novel Thiourea Derivatives Tagged with Thiadiazole, Imidazole and Triazine Moieties as Potential DNA Gyrase and Topoisomerase IV Inhibitors.
Hashem, Heba E; Amr, Abd El-Galil E; Nossier, Eman S; Elsayed, Elsayed A; Azmy, Eman M.
Afiliação
  • Hashem HE; Department of Chemistry, Faculty of Women, Ain Shams University, Heliopolis, Cairo 11457, Egypt.
  • Amr AEE; Drug Exploration & Development Chair (DEDC), Pharmaceutical Chemistry Department, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia.
  • Nossier ES; Applied Organic Chemistry Department, National Research Center, Dokki 12622, Cairo, Egypt.
  • Elsayed EA; Pharmaceutical Medicinal Chemistry Department, Faculty of Pharmacy (Girls), Al-Azhar University, Cairo 11754, Egypt.
  • Azmy EM; Bioproducts Research Chair, Zoology Department, Faculty of Science, King Saud University, Riyadh 11451, Saudi Arabia.
Molecules ; 25(12)2020 Jun 15.
Article em En | MEDLINE | ID: mdl-32549386

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tioureia / DNA Topoisomerase IV / Inibidores da Topoisomerase II Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tioureia / DNA Topoisomerase IV / Inibidores da Topoisomerase II Idioma: En Ano de publicação: 2020 Tipo de documento: Article