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Macrocyclization of a Ligand Targeting a Toxic RNA Dramatically Improves Potency.
Benhamou, Raphael I; Vezina-Dawod, Simon; Choudhary, Shruti; Won Wang, Kye; Meyer, Samantha M; Yildirim, Ilyas; Disney, Matthew D.
Afiliação
  • Benhamou RI; Departments of Chemistry and Neuroscience, The Scripps Research Institute, 130 Scripps Way, Jupiter, FL 33458, USA.
  • Vezina-Dawod S; Departments of Chemistry and Neuroscience, The Scripps Research Institute, 130 Scripps Way, Jupiter, FL 33458, USA.
  • Choudhary S; Departments of Chemistry and Neuroscience, The Scripps Research Institute, 130 Scripps Way, Jupiter, FL 33458, USA.
  • Won Wang K; Department of Chemistry, Florida Atlantic University, John D. MacArthur Campus, Jupiter, FL 33458, USA.
  • Meyer SM; Departments of Chemistry and Neuroscience, The Scripps Research Institute, 130 Scripps Way, Jupiter, FL 33458, USA.
  • Yildirim I; Department of Chemistry, Florida Atlantic University, John D. MacArthur Campus, Jupiter, FL 33458, USA.
  • Disney MD; Departments of Chemistry and Neuroscience, The Scripps Research Institute, 130 Scripps Way, Jupiter, FL 33458, USA.
Chembiochem ; 21(22): 3229-3233, 2020 11 16.
Article em En | MEDLINE | ID: mdl-32649032

Texto completo: 1 Base de dados: MEDLINE Assunto principal: RNA / Bibliotecas de Moléculas Pequenas Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: RNA / Bibliotecas de Moléculas Pequenas Idioma: En Ano de publicação: 2020 Tipo de documento: Article