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Novel Tetrafunctional Probes Identify Target Receptors and Binding Sites of Small-Molecule Drugs from Living Systems.
Miyajima, Rin; Sakai, Koji; Otani, Yuki; Wadatsu, Takashi; Sakata, Yasuyo; Nishikawa, Yuki; Tanaka, Masaki; Yamashita, Yu; Hayashi, Mikayo; Kondo, Kazumi; Hayashi, Takashi.
Afiliação
  • Miyajima R; Medicinal Chemistry Research Laboratories, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Sakai K; Medicinal Chemistry Research Laboratories, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Otani Y; Department of Lead Discovery Research, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Wadatsu T; Department of Lead Discovery Research, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Sakata Y; The Time-Limited Research Project for MSM, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Nishikawa Y; Medicinal Chemistry Research Laboratories, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Tanaka M; Department of Lead Discovery Research, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Yamashita Y; Medicinal Chemistry Research Laboratories, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Hayashi M; Medicinal Chemistry Research Laboratories, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Kondo K; Pharmaceutical Business Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
  • Hayashi T; Department of Lead Discovery Research, New Drug Research Division, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno Kawauchi-cho, Tokushima 771-0192, Japan.
ACS Chem Biol ; 15(9): 2364-2373, 2020 09 18.
Article em En | MEDLINE | ID: mdl-32786265

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tetrazóis / Sondas Moleculares / Receptores de Dopamina D2 / Receptores de GABA / Receptores de AMPA Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Tetrazóis / Sondas Moleculares / Receptores de Dopamina D2 / Receptores de GABA / Receptores de AMPA Idioma: En Ano de publicação: 2020 Tipo de documento: Article