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High affinity rigidified AT2 receptor ligands with indane scaffolds.
Wallinder, Charlotta; Sköld, Christian; Sundholm, Sara; Guimond, Marie-Odile; Yahiaoui, Samir; Lindeberg, Gunnar; Gallo-Payet, Nicole; Hallberg, Mathias; Alterman, Mathias.
Afiliação
  • Wallinder C; Department of Medicinal Chemistry , BMC , Uppsala University , P.O. Box 574 , SE-751 23 Uppsala , Sweden.
  • Sköld C; Department of Medicinal Chemistry , BMC , Uppsala University , P.O. Box 574 , SE-751 23 Uppsala , Sweden.
  • Sundholm S; Department of Medicinal Chemistry , BMC , Uppsala University , P.O. Box 574 , SE-751 23 Uppsala , Sweden.
  • Guimond MO; Service of Endocrinology , Faculty of Medicine and Health Sciences , University of Sherbrooke , Sherbrooke , J1H 5N4 Quebec , Canada.
  • Yahiaoui S; Department of Medicinal Chemistry , BMC , Uppsala University , P.O. Box 574 , SE-751 23 Uppsala , Sweden.
  • Lindeberg G; Department of Medicinal Chemistry , BMC , Uppsala University , P.O. Box 574 , SE-751 23 Uppsala , Sweden.
  • Gallo-Payet N; Service of Endocrinology , Faculty of Medicine and Health Sciences , University of Sherbrooke , Sherbrooke , J1H 5N4 Quebec , Canada.
  • Hallberg M; The Beijer Laboratory , Department of Pharmaceutical Biosciences , Division of Biological Research on Drug Dependence , BMC , Uppsala University , P.O. Box 591 , SE-751 24 Uppsala , Sweden . Email: Mathias.Hallberg@farmbio.uu.se.
  • Alterman M; Department of Medicinal Chemistry , BMC , Uppsala University , P.O. Box 574 , SE-751 23 Uppsala , Sweden.
Medchemcomm ; 10(12): 2146-2160, 2019 Dec 01.
Article em En | MEDLINE | ID: mdl-32904210

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2019 Tipo de documento: Article