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Substituted Azabicyclo[2.2.1]heptanes as Selective Orexin-1 Antagonists: Discovery of JNJ-54717793.
Préville, Cathy; Bonaventure, Pascal; Koudriakova, Tatiana; Lord, Brian; Nepomuceno, Diane; Rizzolio, Michele; Mani, Neelakandha; Coe, Kevin J; Ndifor, Anthony; Dugovic, Christine; Dvorak, Curt A; Coate, Heather; Pippel, Daniel J; Fitzgerald, Anne; Allison, Brett; Lovenberg, Timothy W; Carruthers, Nicholas I; Shireman, Brock T.
Afiliação
  • Préville C; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Bonaventure P; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Koudriakova T; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Lord B; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Nepomuceno D; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Rizzolio M; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Mani N; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Coe KJ; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Ndifor A; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Dugovic C; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Dvorak CA; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Coate H; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Pippel DJ; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Fitzgerald A; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Allison B; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Lovenberg TW; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Carruthers NI; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
  • Shireman BT; Janssen Research & Development L.L.C., 3210 Merryfield Row, San Diego, California 92121, United States.
ACS Med Chem Lett ; 11(10): 2002-2009, 2020 Oct 08.
Article em En | MEDLINE | ID: mdl-33062185

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2020 Tipo de documento: Article