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Synthesis of novel halogenated triarylpyrazoles as selective COX-2 inhibitors: Anti-inflammatory activity, histopatholgical profile and in-silico studies.
Abdellatif, Khaled R A; Abdelall, Eman K A; Labib, Madlen B; Fadaly, Wael A A; Zidan, Taha H.
Afiliação
  • Abdellatif KRA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt; Department of Pharmaceutical Sciences, Ibn Sina National College for Medical Studies, Jeddah, Saudi Arabia.
  • Abdelall EKA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
  • Labib MB; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt. Electronic address: madlen.wanas@pharm.bsu.edu.eg.
  • Fadaly WAA; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
  • Zidan TH; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef 62514, Egypt.
Bioorg Chem ; 105: 104418, 2020 12.
Article em En | MEDLINE | ID: mdl-33166844

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirazóis / Anti-Inflamatórios não Esteroides / Edema / Ciclo-Oxigenase 2 / Inibidores de Ciclo-Oxigenase 2 / Hidrocarbonetos Halogenados Idioma: En Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Pirazóis / Anti-Inflamatórios não Esteroides / Edema / Ciclo-Oxigenase 2 / Inibidores de Ciclo-Oxigenase 2 / Hidrocarbonetos Halogenados Idioma: En Ano de publicação: 2020 Tipo de documento: Article